Published online Aug 16, 2021. doi: 10.12998/wjcc.v9.i23.6929
Peer-review started: May 6, 2021
First decision: June 6, 2021
Revised: June 7, 2021
Accepted: June 22, 2021
Article in press: June 22, 2021
Published online: August 16, 2021
Processing time: 91 Days and 9.5 Hours
Blue rubber bleb naevus syndrome (BRBNS) is a rare disease that usually presents with multiple venous malformations in the skin and gastrointestinal tract. Lesions located in the gastrointestinal tract always result in chronic gastrointestinal bleeding and severe anemia. The successful management of BRBNS with sirolimus had been reported in many institutions, due to its impact on signaling pathways of angiogenesis. However, the experience in treatment of neonates with BRBNS was limited.
A 38-day-old premature female infant born with multiple skin lesions, presented to our center complaining of severe anemia and hematochezia. Laboratory examination demonstrated that hemoglobin was 5.3 g/dL and contrast-enhanced abdominal computed tomography showed multiple low-density space-occupying lesions in the right lobe of the liver. She was diagnosed as having BRBNS based on typical clinical and examination findings. The patient was treated by transfusions twice and hemostatic drugs but symptoms of anemia were difficult to alleviate. A review of BRBNS case reports found that patients had been successfully treated with sirolimus. Then the patient was treated with sirolimus at an average dose of 0.95 mg/m2/d with a target drug level of 10-15 ng/mL. During 28 mo of treatment, the lesion was reduced, hemoglobin returned to normal, and there were no adverse drug reactions.
This case highlights the dosing regimen and plasma concentration in neonates, for the current common empiric dose is high.
Core Tip: Sirolimus is considered as a first-line drug in treating patients with blue rubber bleb naevus syndrome currently. We present herein successful, long-term treatment of blue rubber bleb naevus syndrome with sirolimus in an infant with the youngest age reported. This case highlights two aspects: The recommended doses of 0.1 mg/kg/d resulted in a plasma concentration that was far beyond the expected 10-15 ng/mL in neonates, and a high plasma concentration of more than 20 ng/mL is associated with a great improvement in the condition. Thus, the dosing regimen and plasma concentration are special in neonates.