Published online Sep 6, 2020. doi: 10.12998/wjcc.v8.i17.3841
Peer-review started: May 12, 2020
First decision: May 21, 2020
Revised: June 2, 2020
Accepted: July 30, 2020
Article in press: July 30, 2020
Published online: September 6, 2020
Processing time: 115 Days and 6.4 Hours
Epidermal growth factor receptor (EGFR) tyrosine-kinase inhibitors are widely used for the treatment of non-small-cell lung cancer with EGFR mutations. However, patients with rare, even compound EGFR mutations have different responses to EGFR-tyrosine-kinase inhibitors, which bring uncertainty to clinical treatment.
A 45-year-old female patient presented with a 3-mo history of cough and white sputum without chest pain. Chest computed tomography revealed lung space-occupying lesions and multiple lymphadenectasis. Bronchoscopy and pathology suggested lung adenocarcinoma. Compound variation of EGFR gene (exon 21 L858R/V834L) was detected in both tissue and circulating tumor deoxyribonucleic acid samples. As a result of next-generation sequencing and her family’s wishes, the patient was given oral treatment with icotinib hydrochloride (125 mg/d, tid) from March 21, 2019 and has achieved stable disease for the last 1 year.
Non-small cell lung adenocarcinoma with EGFR L858R/V834L was treated successfully with icotinib, and it may be a new medication treatment option.
Core tip: In non-small cell lung cancer, epidermal growth factor receptor (EGFR) L858R/V834L compound mutation is rare and targeted treatment of this mutation with icotinib has not been reported. In this report, the patient failed to achieve complete or partial response but achieved stable disease. The patient has been in remission for 1 year with no evidence of metastatic nodal disease, and there are signs of continuous remission. So far, the effect of this compound mutation on the efficacy of EGFR tyrosine kinase inhibitors is not clear. It is also unclear which EGFR tyrosine kinase inhibitor is most effective for this variation. This case suggests icotinib may be a possible clinical treatment.