Published online Sep 14, 2021. doi: 10.3748/wjg.v27.i34.5737
Peer-review started: April 15, 2021
First decision: June 23, 2021
Revised: June 30, 2021
Accepted: August 23, 2021
Article in press: August 23, 2021
Published online: September 14, 2021
Processing time: 146 Days and 14.1 Hours
Melatonin plays a central role in the management of circadian rhythm and was identified in the gastrointestinal tract. Epidemiological studies demonstrated that melatonin has oncostatic effects including induction of epigenetic alteration on different types of tumours. The melatonin receptor MT2 encoded by MTNR1B is generally responsible for mediating the downstream effects of melatonin. The expression of MT2 in tumour mucosa is lower than the normal mucosa in patients with colorectal cancer (CRC).
Growing studies have investigated the association between melatonin and CRC carcinogenesis. However, the relationship between MTNR1B gene polymorphisms and CRC sensitivity is not clear. To analyze the effects of MTNR1B gene polymorphisms on CRC prognosis and evaluate the interactions with aberrant promoter methylation of the CDKN2A and MGMT genes will be of great significance.
In our study, we aimed to explore the association between MTNR1B single-nucleotide polymorphism (SNPs) and the 5-year overall survival (OS) of CRC patients. To further assess the interaction between MTNR1B SNPs and CDKN2A and MGMT gene methylation, we examined the relationship between each SNP and the 5-year OS, with data stratified by the methylation status of the CDKN2A and MGMT gene.
Ninety four CRC patients from Taiwan were enrolled to evaluate the association between MTNR1B SNPs, CDKN2A, MGMT gene hypermethylation and 5-year OS. The MTNR1B gene polymorphisms were screened using the Agena MassARRAY platform with iPLEX gold chemistry. The promoter methylation status of CDKN2A and MGMT was assessed using methylation-specific polymerase chain reaction. Associations of the genetic and epigenetic effect and 5-year OS were assessed using the Cox proportional hazards regression model.
In this retrospective cohort study, we found that MTNR1B SNPs was associated with a significantly increased risk of CRC 5-year OS. A strong cumulative effect of the four polymorphisms on CRC prognosis was observed. In stratified analysis, rs1387153, and rs1447352 risk genotype were determined to be associated with 5-year OS in the unmethylation MGMT gene subgroup. In contrast, rs10830963 and rs1447352 risk genotype with hypermethylation CDKN2A gene had a higher risk of death in five years. Four haplotypes of MTNR1B SNPs were also determined to be associated with increased risk of mortality.
This study is one of few reports which demonstrated the association between MTNR1B SNPs and the 5-year OS in patients with CRC. Our data identified these novel genetic biomarkers combined with CDKN2A and MGMT methylation status for the prediction of CRC prognosis, and the findings could be used to individualise the treatment of patients with CRC.
Based on our findings, the novel genetic biomarkers, MTNR1B, combined with CDKN2A and MGMT gene methylation statuses could be a predictive tool for CRC prognosis. The new set of markers may help physicians make treatment decisions based on the prognostic information and would improve the OS of patients with CRC. This study warrant further investigation of the underlying mechanisms related to oncostatic effects of MTNR1B on CRC.