Published online Apr 19, 2024. doi: 10.5498/wjp.v14.i4.563
Peer-review started: October 11, 2023
First decision: December 26, 2023
Revised: January 9, 2024
Accepted: February 28, 2024
Article in press: February 28, 2024
Published online: April 19, 2024
Processing time: 188 Days and 23.7 Hours
Alzheimer’s disease (AD) is a prevalent neurodegenerative disorder characterized by cognitive decline and neuronal loss. Oxidative stress and neuroinflammation play pivotal roles in the pathogenesis of this disease. Tanshinone IIA (Tan-IIA), which is derived from Salvia miltiorrhiza, shows potential neuroprotective effects. Understanding the molecular mechanisms underlying these effects is crucial for the development of novel therapeutic strategies.
The motivation for this study was to elucidate the mechanisms by which Tan-IIA exerts neuroprotective effects in AD, focusing on the potential modulation of the long non-coding RNA (lncRNA) nuclear enriched abundant transcript 1 (NEAT1), microRNA (miR)-291a-3p, and RAB22A, member of the RAS oncogene family (Rab22a) signaling pathways. This has important implications for the development of new AD therapies.
The objective of this study was to investigate the neuroprotective effects of Tan-IIA in AD models and elucidate the underlying molecular mechanisms. Specifically, we aimed to determine how Tan-IIA affects oxidative stress, neuroinflammation, and neuronal viability through the NEAT1/miR-291a-3p/Rab22a signaling axis.
The study employed both in vivo and in vitro models of AD using mice and neural stem cells, respectively. Methods included histopathological examinations, enzyme-linked immunosorbent assays, western blotting, 3-(4,5-dimethylthiazol-2-yl)-2,5-diphenyltetrazolium bromide assays, reverse transcription quantitative polymerase chain reaction assays, and various molecular biology techniques to elucidate the role of the NEAT1/miR-291 a-3p/Rab22a pathway in mediating the effects of Tan-IIA.
Tan-IIA ameliorated AD-related pathological changes, reduced oxidative stress, and attenuated neuroinflammation in the mouse models. It modulated the expression of NEAT1, miR-291a-3p, and Rab22a, indicating the involvement of this signaling axis in its neuroprotective effects. This is the first study to link the amelioration of AD symptoms by Tan-IIA with the downregulation of NEAT1.
Tan-IIA has potential therapeutic roles in AD by attenuating oxidative stress and neuroinflammation, primarily through the NEAT1/miR-291a-3p/Rab22a signaling axis. This highlights the intricate molecular interplay involved in AD and identifies lncRNAs and miRNAs as potential therapeutic targets.
Future research should focus on validating the identified therapeutic targets, namely miR-291a-3p and Rab22a, in clinical AD models. It is also crucial to explore other potential molecular pathways affected by Tan-IIA to fully understand its neuroprotective mechanisms. Clinical trials are essential to determine the efficacy and safety of Tan-IIA-based therapies in patients with AD. Expanding our understanding of the role of NEAT1 in AD could open new avenues for RNA-based therapeutic strategies.