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World J Cardiol. Dec 26, 2014; 6(12): 1245-1251
Published online Dec 26, 2014. doi: 10.4330/wjc.v6.i12.1245
Experimental models of inherited cardiomyopathy and its therapeutics
Miki Nonaka, Sachio Morimoto
Miki Nonaka, Sachio Morimoto, Department of Clinical Pharmacology, Kyushu University Graduate School of Medicine, Fukuoka 812-8582, Japan
Author contributions: Nonaka M wrote the manuscript and designed figures; Morimoto S revised the manuscript and figures; all authors read and approved the final version of the manuscript.
Supported by Grants-in-Aid for Science Research from the Japan Society for the Promotion of Science (JSPS), Nos. 25670130 and 23300145
Correspondence to: Sachio Morimoto, PhD, Department of Clinical Pharmacology, Kyushu University Graduate School of Medicine, 3-1-1 Maidashi, Higashi-ku, Fukuoka 812-8582, Japan. morimoto@med.kyushu-u.ac.jp
Telephone: +81-92-6416081 Fax: +81-92-6426084
Received: May 26, 2014
Revised: July 8, 2014
Accepted: October 14, 2014
Published online: December 26, 2014
Processing time: 216 Days and 12.7 Hours
Abstract

Cardiomyopathy is a disease of myocardium categorized into three major forms, hypertrophic (HCM), dilated (DCM) and restrictive cardiomyopathy (RCM), which has recently been demonstrated to be a monogenic disease due to mutations in various proteins expressed in cardiomyocytes. Mutations in HCM and RCM typically increase the myofilament sensitivity to cytoplasmic Ca2+, leading to systolic hyperfunction and diastolic dysfunction. In contrast, mutations in DCM typically decrease the myofilament sensitivity to cytoplasmic Ca2+ and/or force generation/transmission, leading to systolic dysfunction. Creation of genetically-manipulated transgenic and knock-in animals expressing mutant proteins exogenously and endogenously, respectively, in their hearts provides valuable animal models to discover the molecular and cellular mechanisms for pathogenesis and promising therapeutic strategy in vivo. Recently, cardiomyocytes have been differentiated from patient’s induced pluripotent stem cells as a model of inherited cardiomyopathies in vitro. In this review, we provide overview of experimental models of cardiomyopathies with a focus on revealed molecular and cellular pathogenic mechanisms and potential therapeutics.

Keywords: Cardiomyopathy; Gene; Mutation; Animal model; Induced pluripotent stem cell; Therapeutics

Core tip: Current experimental models of inherited cardiomyopathies (hypertrophic cardiomyopathy, dilated cardiomyopathy and restricted cardiomyopathy), including genetically-manipulated mouse models (transgenic and knock-in mice) and patient’s induced pluripotent stem cell-derived cardiomyocyte models, are summarized and discussed with a focus on revealed molecular pathogenic mechanisms and potential drug therapeutics.