Clinical Research
Copyright ©2008 The WJG Press and Baishideng. All rights reserved.
World J Gastroenterol. Oct 21, 2008; 14(39): 5990-5995
Published online Oct 21, 2008. doi: 10.3748/wjg.14.5990
Rectal administration of d-alpha tocopherol for active ulcerative colitis: A preliminary report
Seyed Amir Mirbagheri, Behtash Ghazi Nezami, Solmaz Assa, Mannan Hajimahmoodi
Seyed Amir Mirbagheri, Behtash Ghazi Nezami, Solmaz Assa, Amir-Alam hospital, Tehran University of Medical Sciences, Tehran 13145-784, Iran
Mannan Hajimahmoodi, Department of Drug and Food Control, Faculty of Pharmacy, Tehran University of Medical Sciences, Tehran 13145-784, Iran
Author contributions: Mirbagheri SA developed the main hypothesis of the study, performed endoscopic studies and clinical examinations, supervised and edited the paper; Mirbagheri SA, Nezami BG, and Assa S designed the research; Nezami BG and Assa S followed the patients and recorded the data; Hajimahmoodi M determined the plasma level of α-tocopherol in recruited patients; Nezami BG and Assa S analyzed the data and wrote the paper.
Supported by Research grant provided by the Tehran University of Medical Sciences
Correspondence to: Seyed Amir Mirbagheri, MD, Depart-ment of Internal Medicine, Amir-Alam Hospital, North Sa’adi Street, Tehran 13145-784, Iran. mirbagherimd@yahoo.com
Telephone: +98-216-6708688 Fax: +98-216-6704805
Received: June 1, 2008
Revised: August 11, 2008
Accepted: August 18, 2008
Published online: October 21, 2008
Abstract

AIM: To investigate the anti-oxidant and anti-neutrophil recruitment effects of rectal d-alpha (d-α) tocopherol administration on mild and moderately active ulcerative colitis (UC).

METHODS: Fifteen patients with mild and moderately active ulcerative colitis were enrolled in an open-label study of d-α tocopherol enema (8000 U/d) for 12 wk. All patients were receiving concomitant therapy with 5-aminosalicylic acid derivatives (5-ASA) and/or immunomodulator medications. Endoscopic evaluation was performed at baseline and after 4th and 12th weeks. Disease activity was measured with the Mayo disease activity index (DAI) and remission was defined as DAI of ≤ 2 with no blood in stool. Clinical response was defined as a DAI reduction of ≥ 2.

RESULTS: At the end of 12th week, the average DAI score significantly decreased compared to the beginning of the study (2.3 ± 0.37 vs 8 ± 0.48, P < 0.0001). One patient was withdrawn after 3 wk for being unavailable to follow-up. On the 4th week of therapy, 12 patients showed clinical response, 3 of whom (21.4%) achieving remission. After 12 wk, all 14 patients responded clinically to the therapy and remission was induced in 9 of them (64%). No patient reported adverse events or was hospitalized due to worsened disease activity.

CONCLUSION: This preliminary report suggests that rectal d-α tocopherol may represent a novel therapy for mild and moderately active UC. The observed results might be due to the anti-inflammatory and anti-oxidative properties of vitamin E.

Keywords: Vitamin E; Ulcerative colitis; Inflammatory bowel disease; Enema; Activity index