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For: Talele TT. Acetylene Group, Friend or Foe in Medicinal Chemistry. J Med Chem 2020;63:5625-63. [PMID: 32031378 DOI: 10.1021/acs.jmedchem.9b01617] [Cited by in Crossref: 23] [Cited by in F6Publishing: 15] [Article Influence: 11.5] [Reference Citation Analysis]
Number Citing Articles
1 Maganti LHB, Ramesh D, Vijayakumar BG, Khan MIK, Dhayalan A, Kamalraja J, Kannan T. Acetylene containing 2-(2-hydrazinyl)thiazole derivatives: design, synthesis, and in vitro and in silico evaluation of antimycobacterial activity against Mycobacterium tuberculosis. RSC Adv 2022;12:8771-82. [PMID: 35424819 DOI: 10.1039/d2ra00928e] [Reference Citation Analysis]
2 Halkina T, Henderson JL, Lin EY, Himmelbauer MK, Jones JH, Nevalainen M, Feng J, King K, Rooney M, Johnson JL, Marcotte DJ, Chodaparambil JV, Kumar PR, Patterson TA, Murugan P, Schuman E, Wong L, Hesson T, Lamore S, Bao C, Calhoun M, Certo H, Amaral B, Dillon GM, Gilfillan R, de Turiso FG. Discovery of Potent and Brain-Penetrant Tau Tubulin Kinase 1 (TTBK1) Inhibitors that Lower Tau Phosphorylation In Vivo. J Med Chem 2021;64:6358-80. [PMID: 33944571 DOI: 10.1021/acs.jmedchem.1c00382] [Reference Citation Analysis]
3 Litti L, Trivini S, Ferraro D, Reguera J. 3D Printed Microfluidic Device for Magnetic Trapping and SERS Quantitative Evaluation of Environmental and Biomedical Analytes. ACS Appl Mater Interfaces 2021;13:34752-61. [PMID: 34256559 DOI: 10.1021/acsami.1c09771] [Reference Citation Analysis]
4 Capaldo L, Ravelli D. Decatungstate as Direct Hydrogen Atom Transfer Photocatalyst for SOMOphilic Alkynylation. Org Lett 2021;23:2243-7. [PMID: 33656899 DOI: 10.1021/acs.orglett.1c00381] [Cited by in Crossref: 13] [Cited by in F6Publishing: 6] [Article Influence: 13.0] [Reference Citation Analysis]
5 Amos SGE, Cavalli D, Le Vaillant F, Waser J. Direct Photoexcitation of Ethynylbenziodoxolones: An Alternative to Photocatalysis for Alkynylation Reactions*. Angew Chem Int Ed Engl 2021;60:23827-34. [PMID: 34403571 DOI: 10.1002/anie.202110257] [Reference Citation Analysis]
6 Pracitto R, Wilcox KC, Lindemann M, Tong J, Zheng C, Li S, Finnema SJ, Huang Y, Cai Z. Further Investigation of Synaptic Vesicle Protein 2A (SV2A) Ligands Designed for Positron Emission Tomography and Single-Photon Emission Computed Tomography Imaging: Synthesis and Structure-Activity Relationship of Substituted Pyridinylmethyl-4-(3,5-difluorophenyl)pyrrolidin-2-ones. ACS Omega 2021;6:27676-83. [PMID: 34722967 DOI: 10.1021/acsomega.1c02433] [Cited by in Crossref: 1] [Article Influence: 1.0] [Reference Citation Analysis]
7 Dombrowski AW, Aguirre AL, Shrestha A, Sarris KA, Wang Y. The Chosen Few: Parallel Library Reaction Methodologies for Drug Discovery. J Org Chem 2021. [PMID: 34780177 DOI: 10.1021/acs.joc.1c01427] [Cited by in Crossref: 1] [Cited by in F6Publishing: 1] [Article Influence: 1.0] [Reference Citation Analysis]
8 Lasso JD, Castillo-Pazos DJ, Li CJ. Green chemistry meets medicinal chemistry: a perspective on modern metal-free late-stage functionalization reactions. Chem Soc Rev 2021. [PMID: 34382989 DOI: 10.1039/d1cs00380a] [Reference Citation Analysis]
9 Li Y, Yang G, Zhang J, Tang P, Yang C, Wang G, Chen J, Liu J, Zhang L, Ouyang L. Discovery, Synthesis, and Evaluation of Highly Selective Vascular Endothelial Growth Factor Receptor 3 (VEGFR3) Inhibitor for the Potential Treatment of Metastatic Triple-Negative Breast Cancer. J Med Chem 2021;64:12022-48. [PMID: 34351741 DOI: 10.1021/acs.jmedchem.1c00678] [Reference Citation Analysis]
10 Fuerst R, Breinbauer R. Activity-Based Protein Profiling (ABPP) of Oxidoreductases. Chembiochem 2021;22:630-8. [PMID: 32881211 DOI: 10.1002/cbic.202000542] [Cited by in Crossref: 1] [Cited by in F6Publishing: 3] [Article Influence: 0.5] [Reference Citation Analysis]
11 Zhang J, Wang M, Wang H, Xu H, Chen J, Guo Z, Ma B, Ban SR, Dai HX. Construction of 2-alkynyl aza-spiro[4,5]indole scaffolds via sequential C-H activations for modular click chemistry libraries. Chem Commun (Camb) 2021;57:8656-9. [PMID: 34373875 DOI: 10.1039/d1cc02798k] [Reference Citation Analysis]
12 Peng X, Xu J, Li T, Chi YR, Jin Z. Chemo-selective cross reaction of two enals via carbene-catalyzed dual activation. Chem Sci 2020;11:12533-9. [PMID: 34123233 DOI: 10.1039/d0sc03297b] [Cited by in Crossref: 2] [Article Influence: 1.0] [Reference Citation Analysis]
13 Song P, Zhao F, Li D, Qu J, Yao M, Su Y, Wang H, Zhou M, Wang Y, Gao Y, Li F, Zhao D, Zhang F, Rao Y, Xia M, Li H, Wang J, Cheng M. Synthesis of selective PAK4 inhibitors for lung metastasis of lung cancer and melanoma cells. Acta Pharmaceutica Sinica B 2022;12:2905-22. [DOI: 10.1016/j.apsb.2022.02.029] [Reference Citation Analysis]
14 Karaj E, Dlamini S, Koranne R, Sindi SH, Perera L, Taylor WR, Viranga Tillekeratne L. Pharmacophore optimization of imidazole chalcones to modulate microtubule dynamics. Bioorganic Chemistry 2022;122:105700. [DOI: 10.1016/j.bioorg.2022.105700] [Reference Citation Analysis]
15 Mishiro K, Nomura M, Furuyama T, Kunishima M. Efficiency Enhancement of a Photocatalytic Decarbonylation of an Aminocyclopropenone by Benzothiophene Substitution. J Org Chem 2021;86:3625-36. [PMID: 33555890 DOI: 10.1021/acs.joc.0c02997] [Reference Citation Analysis]
16 Behroz I, Kleebauer L, Hommernick K, Seidel M, Grätz S, Mainz A, Weston JB, Süssmuth RD. Acetylenic Replacement of Albicidin's Methacrylamide Residue Circumvents Detrimental E/Z Photoisomerization and Preserves Antibacterial Activity. Chemistry 2021;27:9077-86. [PMID: 33769627 DOI: 10.1002/chem.202100523] [Cited by in Crossref: 2] [Cited by in F6Publishing: 2] [Article Influence: 2.0] [Reference Citation Analysis]
17 Wu X, Zhang Y, Liu S, Liu C, Tang G, Cao X, Lei X, Peng J. Research applications of “linkers” in small molecule drugs design in fragment-based. Bioorganic Chemistry 2022. [DOI: 10.1016/j.bioorg.2022.105921] [Reference Citation Analysis]
18 Bandarage UK, Aronov AM, Cao J, Come JH, Cottrell KM, Davies RJ, Giroux S, Jacobs M, Mahajan S, Messersmith D, Moody CS, Swett R, Xu J. Discovery of a Novel Series of Potent and Selective Alkynylthiazole-Derived PI3Kγ Inhibitors. ACS Med Chem Lett 2021;12:129-35. [PMID: 33488974 DOI: 10.1021/acsmedchemlett.0c00573] [Cited by in Crossref: 3] [Cited by in F6Publishing: 3] [Article Influence: 3.0] [Reference Citation Analysis]
19 Li M, Liu T, Li J, He H, Dai H, Xie J. Visible-Light-Mediated Deoxyalkynylation of Activated Tertiary Alcohols. J Org Chem 2021;86:12386-93. [PMID: 34378932 DOI: 10.1021/acs.joc.1c01356] [Cited by in Crossref: 2] [Cited by in F6Publishing: 1] [Article Influence: 2.0] [Reference Citation Analysis]
20 He Q, Zhu L, Yang ZH, Zhu B, Ouyang Q, Du W, Chen YC. Palladium-Catalyzed Modular and Enantioselective cis-Difunctionalization of 1,3-Enynes with Imines and Boronic Reagents. J Am Chem Soc 2021;143:17989-94. [PMID: 34669411 DOI: 10.1021/jacs.1c09877] [Reference Citation Analysis]
21 Chrobak E, Jastrzębska M, Bębenek E, Kadela-Tomanek M, Marciniec K, Latocha M, Wrzalik R, Kusz J, Boryczka S. Molecular Structure, In Vitro Anticancer Study and Molecular Docking of New Phosphate Derivatives of Betulin. Molecules 2021;26:737. [PMID: 33572631 DOI: 10.3390/molecules26030737] [Reference Citation Analysis]
22 Ohno H, Inuki S. Nonbiomimetic total synthesis of indole alkaloids using alkyne-based strategies. Org Biomol Chem 2021;19:3551-68. [PMID: 33908430 DOI: 10.1039/d0ob02577a] [Cited by in Crossref: 2] [Article Influence: 2.0] [Reference Citation Analysis]
23 Zhou T, Jiang MX, Qian PF, Yao QJ, Xu XT, Zhang K, Shi BF. Synthesis of Chiral Sulfoxides via Pd(II)-Catalyzed Enantioselective C-H Alkynylation/Kinetic Resolution of 2-(Arylsulfinyl)pyridines. Org Lett 2021;23:7910-5. [PMID: 34605653 DOI: 10.1021/acs.orglett.1c02918] [Reference Citation Analysis]
24 McHale CM, Karas LJ, Wang X, Wu JI, Miljanić OŠ. Cyclobenzoin Esters as Hosts for Thin Guests. Org Lett 2021;23:2253-7. [PMID: 33635676 DOI: 10.1021/acs.orglett.1c00383] [Reference Citation Analysis]
25 Ponikiewski Ł, Sowa S. Ring Opening of Triflates Derived from Benzophospholan-3-one Oxides by Aryl Grignard Reagents as a Route to 2-Ethynylphenyl(diaryl)phosphine Oxides. J Org Chem 2021;86:14928-41. [PMID: 34699223 DOI: 10.1021/acs.joc.1c01629] [Reference Citation Analysis]
26 Chen D, Xiao Z, Guo H, Gogishvili D, Setroikromo R, van der Wouden PE, Dekker FJ. Identification of a Bromodomain-like Region in 15-Lipoxygenase-1 Explains Its Nuclear Localization. Angew Chem Int Ed Engl 2021. [PMID: 34388301 DOI: 10.1002/anie.202106968] [Reference Citation Analysis]
27 Mons E, Kim RQ, van Doodewaerd BR, van Veelen PA, Mulder MPC, Ovaa H. Exploring the Versatility of the Covalent Thiol-Alkyne Reaction with Substituted Propargyl Warheads: A Deciding Role for the Cysteine Protease. J Am Chem Soc 2021;143:6423-33. [PMID: 33885283 DOI: 10.1021/jacs.0c10513] [Cited by in Crossref: 2] [Cited by in F6Publishing: 1] [Article Influence: 2.0] [Reference Citation Analysis]
28 Yan NL, Santos-Martins D, Nair R, Chu A, Wilson IA, Johnson KA, Forli S, Morgan GJ, Petrassi HM, Kelly JW. Discovery of Potent Coumarin-Based Kinetic Stabilizers of Amyloidogenic Immunoglobulin Light Chains Using Structure-Based Design. J Med Chem 2021;64:6273-99. [PMID: 33939422 DOI: 10.1021/acs.jmedchem.1c00339] [Cited by in Crossref: 1] [Cited by in F6Publishing: 1] [Article Influence: 1.0] [Reference Citation Analysis]
29 Kruszniewska-Rajs C, Strzałka-Mrozik B, Kimsa-Dudek M, Synowiec-Wojtarowicz A, Chrobak E, Bębenek E, Boryczka S, Głuszek S, Gola JM. The Influence of Betulin and Its Derivatives EB5 and ECH147 on the Antioxidant Status of Human Renal Proximal Tubule Epithelial Cells. Int J Mol Sci 2022;23:2524. [PMID: 35269667 DOI: 10.3390/ijms23052524] [Reference Citation Analysis]
30 Bezerra Bellei JC, Glanzmann N, Carpinter BA, Renhe DC, Marques CB, Azevedo MR, Barreto LM, Rocha VN, Karine da Costa Nunes I, Gualberto Pereira HM, Coimbra ES, Ferraz Coelho EA, David da Silva A, de Pilla Varotti F, Gorza Scopel KK. A simple quinoline salt derivative is active in vitro against plasmodium Faciparum asexual blood stages and inhibits the development of cerebral malaria in murine model. Chem Biol Interact 2022;:109848. [PMID: 35149084 DOI: 10.1016/j.cbi.2022.109848] [Reference Citation Analysis]
31 Subbaiah MAM, Meanwell NA. Bioisosteres of the Phenyl Ring: Recent Strategic Applications in Lead Optimization and Drug Design. J Med Chem 2021;64:14046-128. [PMID: 34591488 DOI: 10.1021/acs.jmedchem.1c01215] [Reference Citation Analysis]