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For: Subbaiah MAM, Meanwell NA. Bioisosteres of the Phenyl Ring: Recent Strategic Applications in Lead Optimization and Drug Design. J Med Chem 2021;64:14046-128. [PMID: 34591488 DOI: 10.1021/acs.jmedchem.1c01215] [Cited by in Crossref: 25] [Cited by in F6Publishing: 35] [Article Influence: 25.0] [Reference Citation Analysis]
Number Citing Articles
1 Young RJ, Flitsch SL, Grigalunas M, Leeson PD, Quinn RJ, Turner NJ, Waldmann H. The Time and Place for Nature in Drug Discovery. JACS Au 2022;2:2400-2416. [DOI: 10.1021/jacsau.2c00415] [Reference Citation Analysis]
2 Rigotti T, Bach T. Bicyclo[2.1.1]hexanes by Visible Light-Driven Intramolecular Crossed [2 + 2] Photocycloadditions. Org Lett 2022. [DOI: 10.1021/acs.orglett.2c03606] [Reference Citation Analysis]
3 Li H, Gao Y, Ma J. Advances in nonclassical phenyl bioisosteres for drug structural optimization. Future Medicinal Chemistry 2022;14:1681-1692. [DOI: 10.4155/fmc-2022-0188] [Reference Citation Analysis]
4 Zhang J, Wang T, Qian J, Zhang Y, Zhang J. Ultrasound-promoted three-component halogenation-azaheteroarylation of alkenes involving carbon-halogen and carbon-carbon bond formation. Tetrahedron Letters 2022;110:154198. [DOI: 10.1016/j.tetlet.2022.154198] [Reference Citation Analysis]
5 Yang H, Chen Y, Dang C, Hong AN, Feng P, Bu X. Optimization of Pore-Space-Partitioned Metal–Organic Frameworks Using the Bioisosteric Concept. J Am Chem Soc 2022. [DOI: 10.1021/jacs.2c09349] [Reference Citation Analysis]
6 Liang Y, Kleinmans R, Daniliuc CG, Glorius F. Synthesis of Polysubstituted 2-Oxabicyclo[2.1.1]hexanes via Visible-Light-Induced Energy Transfer. J Am Chem Soc 2022. [DOI: 10.1021/jacs.2c09248] [Reference Citation Analysis]
7 Epplin RC, Paul S, Herter L, Salome C, Hancock EN, Larrow JF, Baum EW, Dunstan DR, Ginsburg-Moraff C, Fessard TC, Brown MK. [2]-Ladderanes as isosteres for meta-substituted aromatic rings and rigidified cyclohexanes. Nat Commun 2022;13:6056. [PMID: 36229621 DOI: 10.1038/s41467-022-33827-3] [Reference Citation Analysis]
8 Turanlı S, Nalbat E, Lengerli D, İbiş K, Güntekin Ergün S, Akhan Güzelcan E, Muyan M, Cetin-atalay R, Çalışkan B, Banoglu E. Vicinal Diaryl-Substituted Isoxazole and Pyrazole Derivatives with In Vitro Growth Inhibitory and In Vivo Antitumor Activity. ACS Omega. [DOI: 10.1021/acsomega.2c03405] [Reference Citation Analysis]
9 Janin YL. On drug discovery against infectious diseases and academic medicinal chemistry contributions. Beilstein J Org Chem 2022;18:1355-78. [DOI: 10.3762/bjoc.18.141] [Reference Citation Analysis]
10 Cossy J, Polàk P, Ruer PC. Incorporation of a cyclobutyl substituent in molecules by transition metal-catalyzed cross-coupling reactions. Org Biomol Chem 2022. [PMID: 36148586 DOI: 10.1039/d2ob01045c] [Reference Citation Analysis]
11 Guo R, Adak S, Bellotti P, Gao X, Smith WW, Le SN, Ma J, Houk KN, Glorius F, Chen S, Brown MK. Photochemical Dearomative Cycloadditions of Quinolines and Alkenes: Scope and Mechanism Studies. J Am Chem Soc . [DOI: 10.1021/jacs.2c07726] [Reference Citation Analysis]
12 Romero-fernández MP, Cintas P, Rojas-buzo S. Switchable Cycloadditions of Mesoionic Dipoles: Refreshing up a Regioselective Approach to Two Distinctive Heterocycles. J Org Chem . [DOI: 10.1021/acs.joc.2c01444] [Reference Citation Analysis]
13 Zhang Y, Li K, Gao W, Liu X, Yuan H, Tang L, Fan Z. Tandem Synthesis of 1,2,3-Thiadiazoles with 3,4-Dichloroisothiazoles and Hydrazines under External Oxidant- and Sulfur-Free Conditions. Org Lett 2022. [PMID: 36054902 DOI: 10.1021/acs.orglett.2c02595] [Cited by in Crossref: 1] [Cited by in F6Publishing: 1] [Article Influence: 1.0] [Reference Citation Analysis]
14 Regueiro-Ren A, Sit SY, Chen Y, Chen J, Swidorski JJ, Liu Z, Venables BL, Sin N, Hartz RA, Protack T, Lin Z, Zhang S, Li Z, Wu DR, Li P, Kempson J, Hou X, Gupta A, Rampulla R, Mathur A, Park H, Sarjeant A, Benitex Y, Rahematpura S, Parker D, Phillips T, Haskell R, Jenkins S, Santone KS, Cockett M, Hanumegowda U, Dicker I, Meanwell NA, Krystal M. The Discovery of GSK3640254, a Next-Generation Inhibitor of HIV-1 Maturation. J Med Chem 2022. [PMID: 36044257 DOI: 10.1021/acs.jmedchem.2c00879] [Cited by in F6Publishing: 2] [Reference Citation Analysis]
15 Salgueiro DC, Chi BK, Guzei IA, García‐reynaga P, Weix DJ. Control of Redox‐Active Ester Reactivity Enables a General Cross‐Electrophile Approach to Access Arylated Strained Rings**. Angew Chem Int Ed 2022;61. [DOI: 10.1002/anie.202205673] [Reference Citation Analysis]
16 Bolduc PN, Pfaffenbach M, Blasczak VD, Mathieu SR, Peterson EA. Synthesis of N-Substituted 3-Amino-2-pyridones. Org Lett 2022. [PMID: 35960821 DOI: 10.1021/acs.orglett.2c02189] [Reference Citation Analysis]
17 Ju H, Hou L, Zhao F, Zhang Y, Jia R, Guizzo L, Bonomini A, Zhang J, Gao Z, Liang R, Bertagnin C, Kong X, Ma X, Kang D, Loregian A, Huang B, Liu X, Zhan P. Iterative Optimization and Structure-Activity Relationship Studies of Oseltamivir Amino Derivatives as Potent and Selective Neuraminidase Inhibitors via Targeting 150-Cavity. J Med Chem 2022. [PMID: 35939763 DOI: 10.1021/acs.jmedchem.1c01970] [Reference Citation Analysis]
18 Ertl P, Altmann E, Racine S, Lewis R. Ring replacement recommender: Ring modifications for improving biological activity. European Journal of Medicinal Chemistry 2022;238:114483. [DOI: 10.1016/j.ejmech.2022.114483] [Reference Citation Analysis]
19 Sousa JLC, Albuquerque HMT, Silvestre AJD, Silva AMS. Decoration of A-Ring of a Lupane-Type Triterpenoid with Different Oxygen and Nitrogen Heterocycles. Molecules 2022;27:4904. [DOI: 10.3390/molecules27154904] [Reference Citation Analysis]
20 Liu K, Zheng W, Chen Y, Tang M, Li D, Deng D, Yang T, Zhang C, Liu J, Yuan X, Shi M, Li X, Guo Y, Zhou Y, Zhao M, Chen L. Discovery, Optimization, and Evaluation of Potent and Selective PI3Kδ-γ Dual Inhibitors for the Treatment of B-cell Malignancies. J Med Chem 2022. [PMID: 35831917 DOI: 10.1021/acs.jmedchem.2c00568] [Reference Citation Analysis]
21 Liu Z, Duan Z, Zhang D, Xiao P, Zhang T, Xu H, Wang CH, Rao GW, Gan J, Huang Y, Yang CG, Dong Z. Structure-Activity Relationships and Antileukemia Effects of the Tricyclic Benzoic Acid FTO Inhibitors. J Med Chem 2022. [PMID: 35793358 DOI: 10.1021/acs.jmedchem.2c00848] [Reference Citation Analysis]
22 Meanwell NA, Loiseleur O. Applications of Isosteres of Piperazine in the Design of Biologically Active Compounds: Part 2. J Agric Food Chem 2022. [PMID: 35675052 DOI: 10.1021/acs.jafc.2c00729] [Cited by in Crossref: 1] [Cited by in F6Publishing: 2] [Article Influence: 1.0] [Reference Citation Analysis]
23 Hill J, Crich D. The N,N,O-Trisubstituted Hydroxylamine Isostere and Its Influence on Lipophilicity and Related Parameters. ACS Med Chem Lett 2022;13:799-806. [PMID: 35586423 DOI: 10.1021/acsmedchemlett.1c00713] [Reference Citation Analysis]
24 Guo R, Chang YC, Herter L, Salome C, Braley SE, Fessard TC, Brown MK. Strain-Release [2π + 2σ] Cycloadditions for the Synthesis of Bicyclo[2.1.1]hexanes Initiated by Energy Transfer. J Am Chem Soc 2022;144:7988-94. [PMID: 35476547 DOI: 10.1021/jacs.2c02976] [Cited by in Crossref: 2] [Cited by in F6Publishing: 7] [Article Influence: 2.0] [Reference Citation Analysis]
25 Escolano M, Cabrera-Afonso MJ, Ribagorda M, Badir SO, Molander GA. Nickel-Mediated Synthesis of Non-Anomeric C-Acyl Glycosides through Electron Donor-Acceptor Complex Photoactivation. J Org Chem 2022. [PMID: 35289617 DOI: 10.1021/acs.joc.1c03041] [Cited by in Crossref: 2] [Cited by in F6Publishing: 2] [Article Influence: 2.0] [Reference Citation Analysis]
26 Naidu BN, Patel M, McAuliffe B, Ding B, Cianci C, Simmermacher J, Jenkins S, Parker DD, Sivaprakasam P, Khan JA, Kish K, Lewis H, Hanumegowda U, Krystal M, Meanwell NA, Kadow JF. Design, Synthesis, and Preclinical Profiling of GSK3739936 (BMS-986180), an Allosteric Inhibitor of HIV-1 Integrase with Broad-Spectrum Activity toward 124/125 Polymorphs. J Med Chem 2022. [PMID: 35235334 DOI: 10.1021/acs.jmedchem.1c02169] [Cited by in Crossref: 4] [Cited by in F6Publishing: 4] [Article Influence: 4.0] [Reference Citation Analysis]
27 Svirčev M, Popsavin M, Pavić A, Vasiljević B, Rodić MV, Djokić S, Kesić J, Srećo Zelenović B, Popsavin V, Kojić V. Design, synthesis, and biological evaluation of thiazole bioisosteres of goniofufurone through in vitro antiproliferative activity and in vivo toxicity. Bioorganic Chemistry 2022. [DOI: 10.1016/j.bioorg.2022.105691] [Cited by in Crossref: 2] [Cited by in F6Publishing: 2] [Article Influence: 2.0] [Reference Citation Analysis]
28 Mills LR, Gygi D, Ludwig JR, Simmons EM, Wisniewski SR, Kim J, Chirik PJ. Cobalt-Catalyzed C(sp 2 )–C(sp 3 ) Suzuki–Miyaura Cross-Coupling Enabled by Well-Defined Precatalysts with L,X-Type Ligands. ACS Catal 2022;12:1905-18. [DOI: 10.1021/acscatal.1c05586] [Cited by in Crossref: 2] [Cited by in F6Publishing: 2] [Article Influence: 2.0] [Reference Citation Analysis]
29 黄 云. Design, Synthesis and Molecular Docking of SARS-CoV-2 3CL<sup>pro</sup> Inhibitors. HJMCe 2022;10:352-357. [DOI: 10.12677/hjmce.2022.104037] [Reference Citation Analysis]
30 Kelly CB, Milligan JA, Tilley LJ, Sodano TM. Bicyclobutanes: from curiosities to versatile reagents and covalent warheads. Chem Sci . [DOI: 10.1039/d2sc03948f] [Cited by in F6Publishing: 1] [Reference Citation Analysis]
31 Li C, Yan H. Recent trends and tactics in facile functionalization of neutral icosahedral carboranes (C2B10H12) and nido-carborane (7,8-C2B9H12−). Advances in Catalysis 2022. [DOI: 10.1016/bs.acat.2022.06.002] [Reference Citation Analysis]
32 Li H, Chen P, Wu Z, Lu Y, Peng J, Chen J, He W. Electrochemical Oxidative Cross-Dehydrogenative Coupling of Five-Membered Aromatic Heterocycles with NH4SCN. Chinese Journal of Organic Chemistry 2022;42:3398. [DOI: 10.6023/cjoc202207009] [Reference Citation Analysis]