BPG is committed to discovery and dissemination of knowledge
Cited by in F6Publishing
For: Talele TT. Opportunities for Tapping into Three-Dimensional Chemical Space through a Quaternary Carbon. J Med Chem 2020;63:13291-315. [PMID: 32805118 DOI: 10.1021/acs.jmedchem.0c00829] [Cited by in Crossref: 13] [Cited by in F6Publishing: 13] [Article Influence: 6.5] [Reference Citation Analysis]
Number Citing Articles
1 Simlandy AK, Lyu MY, Brown MK. Catalytic Arylboration of Spirocyclic Cyclobutenes: Rapid Access to Highly Substituted Spiro[3.n]alkanes. ACS Catal 2021;11:12815-20. [PMID: 35464106 DOI: 10.1021/acscatal.1c03491] [Cited by in Crossref: 6] [Cited by in F6Publishing: 1] [Article Influence: 6.0] [Reference Citation Analysis]
2 Sedenkova KN, Andriasov KS, Eremenko MG, Grishin YK, Alferova VA, Baranova AA, Zefirov NA, Zefirova ON, Zarubaev VV, Gracheva YA, Milaeva ER, Averina EB. Bicyclic Isoxazoline Derivatives: Synthesis and Evaluation of Biological Activity. Molecules 2022;27:3546. [PMID: 35684482 DOI: 10.3390/molecules27113546] [Reference Citation Analysis]
3 Candish L, Collins KD, Cook GC, Douglas JJ, Gómez-Suárez A, Jolit A, Keess S. Photocatalysis in the Life Science Industry. Chem Rev 2021. [PMID: 34558888 DOI: 10.1021/acs.chemrev.1c00416] [Cited by in Crossref: 3] [Article Influence: 3.0] [Reference Citation Analysis]
4 Liu W, Lavagnino MN, Gould CA, Alcázar J, MacMillan DWC. A biomimetic SH2 cross-coupling mechanism for quaternary sp3-carbon formation. Science 2021;374:1258-63. [PMID: 34762491 DOI: 10.1126/science.abl4322] [Reference Citation Analysis]
5 Wang W, Taber DF, Renata H. Practical Enzymatic Production of Carbocycles. Chemistry 2021;27:11773-94. [PMID: 34107092 DOI: 10.1002/chem.202101232] [Reference Citation Analysis]
6 Shirokova VV, Smirnov AY, Zaitseva ER, Baleeva NS, Mikhaylov AА, Baranov MS. Synthesis of julolidine derivatives via SnCl4-promoted spirocyclization of (1-alkyltetrahydroquinolin-8-yl)methylidene-1H-imidazol-5(4H)-ones. Chem Heterocycl Comp. [DOI: 10.1007/s10593-022-03080-z] [Reference Citation Analysis]
7 Pan B, Shi Y, Dong S, He J, Mu B, Wu W, Zhou Y, Zhou F, Zhou J. Highly stereoselective synthesis of spirocyclopropylthiooxindoles and biological evaluation. Org Chem Front 2022;9:2640-6. [DOI: 10.1039/d2qo00300g] [Reference Citation Analysis]
8 Ueda H, Wipf P, Nakamura H. Synthesis of sp3-rich chiral bicyclo[3.3.1]nonanes for chemical space expansion and study of biological activities. Bioorg Med Chem 2021;54:116561. [PMID: 34920311 DOI: 10.1016/j.bmc.2021.116561] [Reference Citation Analysis]
9 Chen WW, Fernández NP, Baranda MD, Cunillera A, Rodríguez LG, Shafir A, Cuenca AB. Exploring benzylic gem-C(sp3)-boron-silicon and boron-tin centers as a synthetic platform. Chem Sci 2021;12:10514-21. [PMID: 34447544 DOI: 10.1039/d1sc01741a] [Reference Citation Analysis]
10 Jung M, Lindsay VNG. One-Pot Synthesis of Strain-Release Reagents from Methyl Sulfones. J Am Chem Soc . [DOI: 10.1021/jacs.2c00923] [Reference Citation Analysis]
11 Asano K. Multipoint Recognition of Molecular Conformations with Organocatalysts for Asymmetric Synthetic Reactions. BCSJ 2021;94:694-712. [DOI: 10.1246/bcsj.20200343] [Cited by in Crossref: 2] [Article Influence: 2.0] [Reference Citation Analysis]
12 Pan A, Chojnacka M, Crowley R 3rd, Göttemann L, Haines BE, Kou KGM. Synergistic Brønsted/Lewis acid catalyzed aromatic alkylation with unactivated tertiary alcohols or di-tert-butylperoxide to synthesize quaternary carbon centers. Chem Sci 2022;13:3539-48. [PMID: 35432882 DOI: 10.1039/d1sc06422c] [Reference Citation Analysis]
13 Peng Y, Huo X, Luo Y, Wu L, Zhang W. Enantio‐ and Diastereodivergent Synthesis of Spirocycles through Dual‐Metal‐Catalyzed [3+2] Annulation of 2‐Vinyloxiranes with Nucleophilic Dipoles. Angew Chem 2021;133:25145-53. [DOI: 10.1002/ange.202111842] [Cited by in Crossref: 9] [Cited by in F6Publishing: 1] [Article Influence: 9.0] [Reference Citation Analysis]
14 Sexton M, Malachowski WP, Yap GPA, Rachii D, Feldman G, Krasley AT, Chen Z, Tran MA, Wiley K, Matei A, Petersen S, Tien ST. Catalytic Enantioselective Birch-Heck Sequence for the Synthesis of Phenanthridinone Derivatives with an All-Carbon Quaternary Stereocenter. J Org Chem 2022;87:1154-72. [PMID: 34985891 DOI: 10.1021/acs.joc.1c02523] [Reference Citation Analysis]
15 Lou SJ, Luo G, Yamaguchi S, An K, Nishiura M, Hou Z. Modular Access to Spiro-dihydroquinolines via Scandium-Catalyzed Dearomative Annulation of Quinolines with Alkynes. J Am Chem Soc 2021;143:20462-71. [PMID: 34813697 DOI: 10.1021/jacs.1c10743] [Cited by in Crossref: 2] [Cited by in F6Publishing: 1] [Article Influence: 2.0] [Reference Citation Analysis]
16 Zhang W, Li L, Li CC. Synthesis of natural products containing highly strained trans-fused bicyclo[3.3.0]octane: historical overview and future prospects. Chem Soc Rev 2021;50:9430-42. [PMID: 34286715 DOI: 10.1039/d0cs01471k] [Reference Citation Analysis]
17 Furiassi L, Tonogai EJ, Hergenrother PJ. Limonin as a Starting Point for the Construction of Compounds with High Scaffold Diversity. Angew Chem 2021;133:16255-64. [DOI: 10.1002/ange.202104228] [Cited by in Crossref: 2] [Cited by in F6Publishing: 2] [Article Influence: 2.0] [Reference Citation Analysis]
18 Lucas SCC, Atkinson SJ, Chung CW, Davis R, Gordon L, Grandi P, Gray JJR, Grimes T, Phillipou A, Preston AG, Prinjha RK, Rioja I, Taylor S, Tomkinson NCO, Wall I, Watson RJ, Woolven J, Demont EH. Optimization of a Series of 2,3-Dihydrobenzofurans as Highly Potent, Second Bromodomain (BD2)-Selective, Bromo and Extra-Terminal Domain (BET) Inhibitors. J Med Chem 2021;64:10711-41. [PMID: 34260229 DOI: 10.1021/acs.jmedchem.1c00344] [Reference Citation Analysis]
19 Sakai HA, MacMillan DWC. Nontraditional Fragment Couplings of Alcohols and Carboxylic Acids: C(sp3)-C(sp3) Cross-Coupling via Radical Sorting. J Am Chem Soc 2022. [PMID: 35353531 DOI: 10.1021/jacs.2c02062] [Cited by in Crossref: 8] [Cited by in F6Publishing: 5] [Article Influence: 8.0] [Reference Citation Analysis]
20 Lv XY, Abrams R, Martin R. Dihydroquinazolinones as adaptative C(sp3) handles in arylations and alkylations via dual catalytic C-C bond-functionalization. Nat Commun 2022;13:2394. [PMID: 35504911 DOI: 10.1038/s41467-022-29984-0] [Reference Citation Analysis]
21 Chen ZH, Sun RZ, Yao F, Hu XD, Xiang LX, Cong H, Liu WB. Enantioselective Nickel-Catalyzed Reductive Aryl/Alkenyl-Cyano Cyclization Coupling to All-Carbon Quaternary Stereocenters. J Am Chem Soc 2022. [PMID: 35263101 DOI: 10.1021/jacs.2c01237] [Cited by in Crossref: 1] [Article Influence: 1.0] [Reference Citation Analysis]
22 Tyler JL, Noble A, Aggarwal VK. Strain-Release-Driven Friedel-Crafts Spirocyclization of Azabicyclo[1.1.0]butanes. Angew Chem Int Ed Engl 2021. [PMID: 34780681 DOI: 10.1002/anie.202114235] [Reference Citation Analysis]
23 Lou Y, Wei J, Li M, Zhu Y. Distal Ionic Substrate-Catalyst Interactions Enable Long-Range Stereocontrol: Access to Remote Quaternary Stereocenters through a Desymmetrizing Suzuki-Miyaura Reaction. J Am Chem Soc 2022;144:123-9. [PMID: 34979078 DOI: 10.1021/jacs.1c12345] [Cited by in Crossref: 7] [Cited by in F6Publishing: 3] [Article Influence: 7.0] [Reference Citation Analysis]
24 Peil S, Gutiérrez González A, Leutzsch M, Fürstner A. C-H Insertion via Ruthenium Catalyzed gem-Hydrogenation of 1,3-Enynes. J Am Chem Soc 2022. [PMID: 35170941 DOI: 10.1021/jacs.1c13446] [Cited by in Crossref: 8] [Cited by in F6Publishing: 2] [Article Influence: 8.0] [Reference Citation Analysis]
25 Tian Y, Wu F, Jia S, Gong X, Mao H, Wang P, Qin W, Yan H. Organocatalytic Asymmetric Construction of Tetrasubstituted Carbon Stereocenters Bearing Three Heteroatoms via Intramolecular Cyclization of Vinylidene ortho-Quinone Methide with Imidates. Org Lett 2022. [PMID: 35819168 DOI: 10.1021/acs.orglett.2c01842] [Reference Citation Analysis]
26 Liu XL, Li L, Lin HZ, Deng JT, Zhang XZ, Peng JB. Copper-catalyzed 1,2-Borylacylation of 1,3-Enynes: synthesis of β-Alkynyl ketones. Chem Commun (Camb) 2022;58:5968-71. [PMID: 35475443 DOI: 10.1039/d2cc01732f] [Reference Citation Analysis]
27 Malone JA, Philkhana SC, Stepherson JR, Badmus FO, Fronczek FR, Kartika R. Copper(I)-Catalyzed Synthesis of Unsymmetrical All-Carbon Bis-Quaternary Centers at the Opposing α-Carbons of Cyclohexanones. Org Lett 2022. [PMID: 35767696 DOI: 10.1021/acs.orglett.2c01890] [Reference Citation Analysis]
28 Ivanov DS, Zaitseva ER, Smirnov AY, Rustamova DA, Mikhaylov AA, Sycheva MA, Gluschenko DA, Baleeva NS, Baranov MS. Chemodivergent Spirocyclization of 2‐Sec‐Aminobenzilidene Imidazolones: Lewis Versus Brønsted Acids Catalysis. Adv Synth Catal 2022;364:1587-95. [DOI: 10.1002/adsc.202200109] [Reference Citation Analysis]
29 Hiesinger K, Dar'in D, Proschak E, Krasavin M. Spirocyclic Scaffolds in Medicinal Chemistry. J Med Chem 2021;64:150-83. [PMID: 33381970 DOI: 10.1021/acs.jmedchem.0c01473] [Cited by in Crossref: 15] [Cited by in F6Publishing: 12] [Article Influence: 7.5] [Reference Citation Analysis]
30 Modak A, Alegre-Requena JV, de Lescure L, Rynders KJ, Paton RS, Race NJ. Homologation of Electron-Rich Benzyl Bromide Derivatives via Diazo C-C Bond Insertion. J Am Chem Soc 2021. [PMID: 34898193 DOI: 10.1021/jacs.1c11503] [Reference Citation Analysis]
31 Serafini M, Cargnin S, Massarotti A, Tron GC, Pirali T, Genazzani AA. What's in a Name? Drug Nomenclature and Medicinal Chemistry Trends using INN Publications. J Med Chem 2021;64:4410-29. [PMID: 33847110 DOI: 10.1021/acs.jmedchem.1c00181] [Reference Citation Analysis]
32 Sohtome Y, Kanomata K, Sodeoka M. Cross-Coupling Reactions of Persistent Tertiary Carbon Radicals. BCSJ 2021;94:1066-79. [DOI: 10.1246/bcsj.20200376] [Cited by in Crossref: 3] [Cited by in F6Publishing: 3] [Article Influence: 3.0] [Reference Citation Analysis]
33 Peng Y, Huo X, Luo Y, Wu L, Zhang W. Enantio- and Diastereodivergent Synthesis of Spirocycles through Dual-Metal-Catalyzed [3+2] Annulation of 2-Vinyloxiranes with Nucleophilic Dipoles. Angew Chem Int Ed Engl 2021;60:24941-9. [PMID: 34532948 DOI: 10.1002/anie.202111842] [Reference Citation Analysis]
34 Laidlaw G, Franckevičius V. Palladium-Catalyzed Decarboxylative Asymmetric Allylic Alkylation of Thietane 1,1-Dioxides. Org Lett 2021. [PMID: 34914384 DOI: 10.1021/acs.orglett.1c04075] [Reference Citation Analysis]
35 Zhu X, Li R, Yao H, Lin A. Palladium-Catalyzed Allenamide Carbopalladation/Allylation with Active Methine Compounds. Org Lett 2021;23:4630-4. [PMID: 34048265 DOI: 10.1021/acs.orglett.1c01369] [Cited by in Crossref: 1] [Article Influence: 1.0] [Reference Citation Analysis]
36 Pan Y, Ren W, Zhang Z, Luo F, Hou X, Li X, Yang Y, Wang Y. Tandem 1,6-addition/cyclopropanation/rearrangement reaction of vinylogous para -quinone methides with 3-chlorooxindoles: construction of vicinal quaternary carbon centers. Org Chem Front . [DOI: 10.1039/d2qo00471b] [Reference Citation Analysis]
37 Caló FP, Zimmer A, Bistoni G, Fürstner A. From Serendipity to Rational Design: Heteroleptic Dirhodium Amidate Complexes for Diastereodivergent Asymmetric Cyclopropanation. J Am Chem Soc 2022. [PMID: 35420801 DOI: 10.1021/jacs.2c02258] [Cited by in Crossref: 1] [Cited by in F6Publishing: 1] [Article Influence: 1.0] [Reference Citation Analysis]
38 Soklou KE, Marzag H, Vallée B, Routier S, Plé K. Synthesis of Heterospirocycles through Gold‐(I) Catalysis: Useful Building Blocks for Medicinal Chemistry. Adv Synth Catal 2022;364:218-24. [DOI: 10.1002/adsc.202101080] [Cited by in Crossref: 1] [Article Influence: 1.0] [Reference Citation Analysis]
39 Wang M, Li B, Gong B, Yao H, Lin A. Synthesis of pyranopyrazoles with a chiral quaternary carbon stereocenter via copper-catalyzed enantioselective [3 + 3] cycloaddition. Chem Commun (Camb) 2022;58:2850-3. [PMID: 35129569 DOI: 10.1039/d1cc07058d] [Reference Citation Analysis]
40 Morimoto J, Miyamoto K, Ichikawa Y, Uchiyama M, Makishima M, Hashimoto Y, Ishikawa M. Improvement in aqueous solubility of achiral symmetric cyclofenil by modification to a chiral asymmetric analog. Sci Rep 2021;11:12697. [PMID: 34135380 DOI: 10.1038/s41598-021-92028-y] [Reference Citation Analysis]
41 Furiassi L, Tonogai EJ, Hergenrother PJ. Limonin as a Starting Point for the Construction of Compounds with High Scaffold Diversity. Angew Chem Int Ed Engl 2021;60:16119-28. [PMID: 33973348 DOI: 10.1002/anie.202104228] [Cited by in Crossref: 2] [Cited by in F6Publishing: 2] [Article Influence: 2.0] [Reference Citation Analysis]
42 Liu L, Zhou C, Wang C. Construction of highly congested quaternary carbon centers by NHC catalysis through dearomatization. Green Synthesis and Catalysis 2022. [DOI: 10.1016/j.gresc.2022.05.010] [Reference Citation Analysis]
43 Sakai K, Oisaki K, Kanai M. A Germanium Catalyst Accelerates the Photoredox α-C(sp3)-H Alkylation of Primary Amines. Org Lett 2022. [PMID: 35486160 DOI: 10.1021/acs.orglett.2c00871] [Reference Citation Analysis]
44 Fairchild ME, Noble A, Aggarwal VK. Diastereodivergent Synthesis of Cyclopentyl Boronic Esters Bearing Contiguous Fully Substituted Stereocenters. Angewandte Chemie. [DOI: 10.1002/ange.202205816] [Reference Citation Analysis]
45 Giustiniano M, Gruber CW, Kent CN, Trippier PC. Back to the Medicinal Chemistry Future. J Med Chem 2021;64:15515-8. [PMID: 34719927 DOI: 10.1021/acs.jmedchem.1c01788] [Reference Citation Analysis]
46 Doyle MGJ, Gabbey AL, McNutt W, Lundgren RJ. Enantioselective Tertiary Electrophile (Hetero)Benzylation: Pd-Catalyzed Substitution of Isoprene Monoxide with Arylacetates*. Angew Chem Int Ed Engl 2021. [PMID: 34658132 DOI: 10.1002/anie.202110525] [Reference Citation Analysis]
47 Wang L, Han H, Gu L, Zhang W, Zhao J, Wang Q. Skeletal remodeling of chalcone-based pyridinium salts to access isoindoline polycycles and their bridged derivatives. Chem Sci 2021;12:15389-98. [PMID: 34976360 DOI: 10.1039/d1sc05741c] [Cited by in Crossref: 5] [Cited by in F6Publishing: 3] [Article Influence: 5.0] [Reference Citation Analysis]
48 Tsuji T, Hashiguchi K, Yoshida M, Ikeda T, Koga Y, Honda Y, Tanaka T, Re S, Mizuguchi K, Takahashi D, Yazaki R, Ohshima T. α-Amino acid and peptide synthesis using catalytic cross-dehydrogenative coupling. Nat Synth 2022;1:304-12. [DOI: 10.1038/s44160-022-00037-0] [Cited by in Crossref: 4] [Cited by in F6Publishing: 1] [Article Influence: 4.0] [Reference Citation Analysis]
49 Doyle MGJ, Gabbey AL, Mcnutt W, Lundgren RJ. Enantioselective Tertiary Electrophile (Hetero)Benzylation: Pd‐Catalyzed Substitution of Isoprene Monoxide with Arylacetates**. Angew Chem 2021;133:26699-703. [DOI: 10.1002/ange.202110525] [Cited by in Crossref: 2] [Cited by in F6Publishing: 1] [Article Influence: 2.0] [Reference Citation Analysis]
50 Zhang D, Li M, Li J, Lin A, Yao H. Rhodium-catalyzed intermolecular enantioselective Alder-ene type reaction of cyclopentenes with silylacetylenes. Nat Commun 2021;12:6627. [PMID: 34785658 DOI: 10.1038/s41467-021-26955-9] [Reference Citation Analysis]
51 Gao Y, Qin W, Tian M, Zhao X, Hu X. Defluorinative Alkylation of Trifluoromethyl Alkenes with Soft Carbon Nucleophiles Enabled by a Catalytic Amount of Base. Adv Synth Catal. [DOI: 10.1002/adsc.202200328] [Reference Citation Analysis]
52 Dorsheimer JR, Ashley MA, Rovis T. Dual Nickel/Photoredox-Catalyzed Deaminative Cross-Coupling of Sterically Hindered Primary Amines. J Am Chem Soc 2021;143:19294-9. [PMID: 34767360 DOI: 10.1021/jacs.1c10150] [Reference Citation Analysis]
53 Bavo F, de-Jong H, Petersen J, Falk-Petersen CB, Löffler R, Sparrow E, Rostrup F, Eliasen JN, Wilhelmsen KS, Barslund K, Bundgaard C, Nielsen B, Kristiansen U, Wellendorph P, Bogdanov Y, Frølund B. Structure-Activity Studies of 3,9-Diazaspiro[5.5]undecane-Based γ-Aminobutyric Acid Type A Receptor Antagonists with Immunomodulatory Effect. J Med Chem 2021;64:17795-812. [PMID: 34908407 DOI: 10.1021/acs.jmedchem.1c00290] [Reference Citation Analysis]
54 López L, Cabal MP, Valdés C. Construction of NH-Unprotected Spiropyrrolidines and Spiroisoindolines by [4+1] Cyclizations of γ-Azidoboronic Acids with Cyclic N-Sulfonylhydrazones. Angew Chem Int Ed Engl 2021. [PMID: 34677906 DOI: 10.1002/anie.202113370] [Reference Citation Analysis]
55 Yang Y, Tsien J, Ben David A, Hughes JME, Merchant RR, Qin T. Practical and Modular Construction of C(sp3)-Rich Alkyl Boron Compounds. J Am Chem Soc 2021;143:471-80. [PMID: 33347297 DOI: 10.1021/jacs.0c11964] [Cited by in Crossref: 6] [Cited by in F6Publishing: 3] [Article Influence: 3.0] [Reference Citation Analysis]
56 Nagano T, Matsumoto A, Yoshizaki R, Asano K, Matsubara S. Non-enzymatic catalytic asymmetric cyanation of acylsilanes. Commun Chem 2022;5. [DOI: 10.1038/s42004-022-00662-y] [Reference Citation Analysis]
57 Yang Y, Tsien J, Hughes JME, Peters BK, Merchant RR, Qin T. An intramolecular coupling approach to alkyl bioisosteres for the synthesis of multisubstituted bicycloalkyl boronates. Nat Chem 2021;13:950-5. [PMID: 34584254 DOI: 10.1038/s41557-021-00786-z] [Cited by in Crossref: 1] [Article Influence: 1.0] [Reference Citation Analysis]
58 Dampalla CS, Rathnayake AD, Galasiti Kankanamalage AC, Kim Y, Perera KD, Nguyen HN, Miller MJ, Madden TK, Picard HR, Thurman HA, Kashipathy MM, Liu L, Battaile KP, Lovell S, Chang KO, Groutas WC. Structure-Guided Design of Potent Spirocyclic Inhibitors of Severe Acute Respiratory Syndrome Coronavirus-2 3C-like Protease. J Med Chem 2022. [PMID: 35638577 DOI: 10.1021/acs.jmedchem.2c00224] [Reference Citation Analysis]