BPG is committed to discovery and dissemination of knowledge
Cited by in F6Publishing
For: Han J, Remete AM, Dobson LS, Kiss L, Izawa K, Moriwaki H, Soloshonok VA, O’hagan D. Next generation organofluorine containing blockbuster drugs. Journal of Fluorine Chemistry 2020;239:109639. [DOI: 10.1016/j.jfluchem.2020.109639] [Cited by in Crossref: 48] [Cited by in F6Publishing: 12] [Article Influence: 24.0] [Reference Citation Analysis]
Number Citing Articles
1 Amaye IJ, Harper T, L Jackson-ayotunde P. Design and development of trifluoromethylated enaminone derivatives as potential anticonvulsants. Journal of Fluorine Chemistry 2021;251:109886. [DOI: 10.1016/j.jfluchem.2021.109886] [Reference Citation Analysis]
2 Carvalho DR, Christian AH. Modern approaches towards the synthesis of geminal difluoroalkyl groups. Org Biomol Chem 2021;19:947-64. [PMID: 33406177 DOI: 10.1039/d0ob02374d] [Cited by in Crossref: 6] [Article Influence: 6.0] [Reference Citation Analysis]
3 Tyumentsev IA, Kobelevskaya VA, Ushakov IA, Rulev AY. Nucleophilic reactions of ethyl (Z)-2‑bromo-4,4,4-trifluorobut-2-enoate: One molecule – various heterocycles. Journal of Fluorine Chemistry 2022;254:109946. [DOI: 10.1016/j.jfluchem.2021.109946] [Cited by in Crossref: 1] [Cited by in F6Publishing: 1] [Article Influence: 1.0] [Reference Citation Analysis]
4 Sanchez CA, Gadais C, Chaume G, Girard S, Chelain E, Brigaud T. Enantiopure 5-CF3-Proline: Synthesis, Incorporation in Peptides, and Tuning of the Peptide Bond Geometry. Org Lett 2021;23:382-7. [PMID: 33369434 DOI: 10.1021/acs.orglett.0c03880] [Cited by in Crossref: 3] [Cited by in F6Publishing: 1] [Article Influence: 3.0] [Reference Citation Analysis]
5 Benke Z, Nonn M, Remete AM, Fustero S, Kiss L. Diversity-Oriented Synthesis of Highly Functionalized Alicycles across Dipolar Cycloaddition/Metathesis Reaction. Synlett 2021;32:1911-33. [DOI: 10.1055/s-0040-1706041] [Cited by in Crossref: 1] [Cited by in F6Publishing: 1] [Article Influence: 1.0] [Reference Citation Analysis]
6 Chicas-Baños DF, Frontana-Uribe BA. Electrochemical Generation and Use in Organic Synthesis of C-, O-, and N-Centered Radicals. Chem Rec 2021;21:2538-73. [PMID: 34047059 DOI: 10.1002/tcr.202100056] [Reference Citation Analysis]
7 Meyer S, Häfliger J, Schäfer M, Molloy JJ, Daniliuc CG, Gilmour R. Eine chirale pentafluorierte Isopropylgruppe durch Iod(I)/(III)‐Katalyse. Angew Chem 2021;133:6501-6. [DOI: 10.1002/ange.202015946] [Cited by in Crossref: 4] [Cited by in F6Publishing: 1] [Article Influence: 4.0] [Reference Citation Analysis]
8 Urner LM, Young Lee G, Treacy JW, Turlik A, Khan SI, Houk KN, Jung ME. Intramolecular N-H⋅⋅⋅F Hydrogen Bonding Interaction in a Series of 4-Anilino-5-Fluoroquinazolines: Experimental and Theoretical Characterization of Electronic and Conformational Effects. Chemistry 2021. [PMID: 34767667 DOI: 10.1002/chem.202103135] [Reference Citation Analysis]
9 Li W, Kitamura T, Zhou Y, Butler G, Han J, Soloshonok VA. Electrophilic fluorination using PhIO/HF·THF reagent. Journal of Fluorine Chemistry 2020;240:109670. [DOI: 10.1016/j.jfluchem.2020.109670] [Cited by in Crossref: 2] [Cited by in F6Publishing: 1] [Article Influence: 1.0] [Reference Citation Analysis]
10 Kumar T, Yang Y, Sghaier S, Zaid Y, Le Goff XF, Rousset E, Massicot F, Harakat D, Martinez A, Taillefer M, Maron L, Behr J, Jaroschik F. Tuning the Regioselective Functionalization of Trifluoromethylated Dienes via Lanthanum‐Mediated Single C−F Bond Activation. Chem Eur J 2021;27:4016-21. [DOI: 10.1002/chem.202005239] [Cited by in Crossref: 2] [Cited by in F6Publishing: 1] [Article Influence: 2.0] [Reference Citation Analysis]
11 Heard DM, Doobary S, Lennox AJJ. 3D Printed Reactionware for Synthetic Electrochemistry with Hydrogen Fluoride Reagents. ChemElectroChem 2021;8:2070-4. [DOI: 10.1002/celc.202100496] [Cited by in Crossref: 2] [Cited by in F6Publishing: 1] [Article Influence: 2.0] [Reference Citation Analysis]
12 Hao Y, Gong Y, Zhou Y, Zhou J, Yu J. Construction of β-Quaternary α,α-Difluoroketones via Catalytic Nucleophilic Substitution of Tertiary Alcohols with Difluoroenoxysilanes. Org Lett 2020;22:8516-21. [DOI: 10.1021/acs.orglett.0c03123] [Cited by in Crossref: 7] [Cited by in F6Publishing: 4] [Article Influence: 3.5] [Reference Citation Analysis]
13 Sittihan S, Sopha P, Ruchirawat S. Synthesis and Anticancer Activity of Pentafluorobenzenesulfonamide Derivatives as Caspase-Dependent Apoptosis-Inducing Agents. ChemMedChem 2021. [PMID: 34784449 DOI: 10.1002/cmdc.202100637] [Reference Citation Analysis]
14 Dix S, Golz P, Schmid JR, Riedel S, Hopkinson MN. Radical C-H Trifluoromethoxylation of (Hetero)arenes with Bis(trifluoromethyl)peroxide. Chemistry 2021;27:11554-8. [PMID: 34096651 DOI: 10.1002/chem.202101621] [Cited by in Crossref: 1] [Cited by in F6Publishing: 1] [Article Influence: 1.0] [Reference Citation Analysis]
15 Grollier K, Chefdeville E, De Zordo-banliat A, Pegot B, Dagousset G, Magnier E, Billard T. Fe-mediated nucleophilic trifluoromethylselenolation of activated alkyl bromides via umpolung reactivity of trifluoromethyl tolueneselenosulfinate. Tetrahedron 2021;100:132498. [DOI: 10.1016/j.tet.2021.132498] [Reference Citation Analysis]
16 Remete AM, Nonn M, Escorihuela J, Fustero S, Kiss L. Asymmetric Methods for Carbon‐Fluorine Bond Formation. Eur J Org Chem 2021;2021:5946-74. [DOI: 10.1002/ejoc.202101094] [Cited by in Crossref: 2] [Cited by in F6Publishing: 2] [Article Influence: 2.0] [Reference Citation Analysis]
17 Wang T, Li Z, Hu J, Wu T. Copper catalyzed hydrodefluorination of propargylic gem-difluorides with “triple bonds migration”. Tetrahedron 2022. [DOI: 10.1016/j.tet.2022.132897] [Reference Citation Analysis]
18 Pliego JR. Copper-Mediated Aromatic Fluorination Using N-Heterocycle-Carbene Ligand: Free Energy Profile of the Cu(I)/Cu(III) and Cu(II) radical Mechanisms. Journal of Organometallic Chemistry 2022. [DOI: 10.1016/j.jorganchem.2022.122397] [Cited by in Crossref: 1] [Article Influence: 1.0] [Reference Citation Analysis]
19 Zou Y, Takeda R, Han J, Konno H, Moriwaki H, Abe H, Izawa K, Soloshonok VA. Asymmetric Synthesis of N ‐Fmoc‐( S )‐7‐aza‐tryptophan via Alkylation of Chiral Nucleophilic Glycine Equivalent. Eur J Org Chem 2021;2021:2962-5. [DOI: 10.1002/ejoc.202100485] [Cited by in Crossref: 1] [Cited by in F6Publishing: 1] [Article Influence: 1.0] [Reference Citation Analysis]
20 Kaźmierczak M, Bilska‐markowska M. Diethylaminosulfur Trifluoride (DAST) Mediated Transformations Leading to Valuable Building Blocks and Bioactive Compounds. Eur J Org Chem 2021;2021:5585-604. [DOI: 10.1002/ejoc.202101027] [Cited by in Crossref: 3] [Cited by in F6Publishing: 2] [Article Influence: 3.0] [Reference Citation Analysis]
21 Edilova YO, Kudyakova YS, Kiskin MA, Burgart YV, Saloutin VI, Bazhin DN. Expanding 1,2,4-triketone toolbox for use as fluorinated building blocks in the synthesis of pyrazoles, pyridazinones and β-diketohydrazones. Journal of Fluorine Chemistry 2022;253:109932. [DOI: 10.1016/j.jfluchem.2021.109932] [Reference Citation Analysis]
22 Ouchakour L, Nonn M, Remete AM, Kiss L. An Improved Stereocontrolled Access Route to Piperidine or Azepane β‐Amino Esters and Azabicyclic β‐ and γ‐Lactams; Synthesis of Novel Functionalized Azaheterocyles. Eur J Org Chem 2021;2021:3874-85. [DOI: 10.1002/ejoc.202100540] [Cited by in Crossref: 1] [Cited by in F6Publishing: 2] [Article Influence: 1.0] [Reference Citation Analysis]
23 Li S, Lv X, Ren J, Feng L, Ma C. A Direct Method for Synthesis of Fluorinated Quinazolinones and Quinoxalines Using Fluorinated Acids without Metals or Additives. Synthesis. [DOI: 10.1055/a-1824-6352] [Reference Citation Analysis]
24 Wang Q, Zhang X, Sorochinsky AE, Butler G, Han J, Soloshonok VA. Advances in the Development of Trifluoromethoxylation Reagents. Symmetry 2021;13:2380. [DOI: 10.3390/sym13122380] [Cited by in Crossref: 2] [Cited by in F6Publishing: 2] [Article Influence: 2.0] [Reference Citation Analysis]
25 Zemtsov AA, Levin VV, Dilman AD. Allylic substitution reactions with fluorinated nucleophiles. Coordination Chemistry Reviews 2022;459:214455. [DOI: 10.1016/j.ccr.2022.214455] [Reference Citation Analysis]
26 Sun L, Yu Z, Luo X, Ma M, Shen Z, Chu X. Transition-metal-free hydroamination/defluorination/cyclization of perfluoroalkyl alkynes with amidines. Org Chem Front 2021;9:109-16. [DOI: 10.1039/d1qo01439k] [Cited by in Crossref: 6] [Cited by in F6Publishing: 3] [Article Influence: 6.0] [Reference Citation Analysis]
27 Yu Y, Liu A, Dhawan G, Mei H, Zhang W, Izawa K, Soloshonok VA, Han J. Fluorine-containing pharmaceuticals approved by the FDA in 2020: Synthesis and biological activity. Chinese Chemical Letters 2021;32:3342-54. [DOI: 10.1016/j.cclet.2021.05.042] [Cited by in Crossref: 9] [Cited by in F6Publishing: 5] [Article Influence: 9.0] [Reference Citation Analysis]
28 Han J, Konno H, Sato T, Soloshonok VA, Izawa K. Tailor-made amino acids in the design of small-molecule blockbuster drugs. Eur J Med Chem 2021;220:113448. [PMID: 33906050 DOI: 10.1016/j.ejmech.2021.113448] [Cited by in Crossref: 5] [Cited by in F6Publishing: 4] [Article Influence: 5.0] [Reference Citation Analysis]
29 Grollier K, De Zordo‐banliat A, Bourdreux F, Pegot B, Dagousset G, Magnier E, Billard T. (Trifluoromethylselenyl)methylchalcogenyl as Emerging Fluorinated Groups: Synthesis under Photoredox Catalysis and Determination of the Lipophilicity. Chem Eur J 2021;27:6028-33. [DOI: 10.1002/chem.202100053] [Cited by in Crossref: 6] [Cited by in F6Publishing: 1] [Article Influence: 6.0] [Reference Citation Analysis]
30 Zemtsov AA, Lunkov SS, Levin VV, Dilman AD. Synthesis of Trifluoromethylated Dithiocarbamates via Photocatalyzed Substitution Reaction: Pentafluoropyridine as Activating Reagent. Eur J Org Chem 2021;2021:1007-10. [DOI: 10.1002/ejoc.202001572] [Cited by in Crossref: 3] [Cited by in F6Publishing: 1] [Article Influence: 3.0] [Reference Citation Analysis]
31 Motornov VA, Tabolin AA, Nelyubina YV, Nenajdenko VG, Ioffe SL. Copper-catalyzed [3 + 2]-cycloaddition of α-halonitroalkenes with azomethine ylides: facile synthesis of multisubstituted pyrrolidines and pyrroles. Org Biomol Chem 2021;19:3413-27. [PMID: 33899878 DOI: 10.1039/d1ob00146a] [Cited by in Crossref: 3] [Article Influence: 3.0] [Reference Citation Analysis]
32 Häfliger J, Sokolova OO, Lenz M, Daniliuc CG, Gilmour R. Stereokontrollierte Synthese von fluorierten Isochromanen durch Iod(I)/Iod(III)‐Katalyse. Angewandte Chemie. [DOI: 10.1002/ange.202205277] [Reference Citation Analysis]
33 Murtaza A, Qamar MA, Saleem K, Hardwick T, Zia Ul Haq, Shirinfar B, Ahmed N. Renewable Electricity Enables Green Routes to Fine Chemicals and Pharmaceuticals. Chem Rec 2022;:e202100296. [PMID: 35103382 DOI: 10.1002/tcr.202100296] [Cited by in Crossref: 1] [Article Influence: 1.0] [Reference Citation Analysis]
34 Nonn M, Paizs C, Kiss L. Recent Progress in the Selective Fluorinations of Some Functionalized Cycloalkenes. Chem Rec 2022;:e202200130. [PMID: 35680609 DOI: 10.1002/tcr.202200130] [Reference Citation Analysis]
35 Logvinenko IG, Kondratov IS, Dobrydnev AV, Kozytskiy AV, Grygorenko OO. Synthesis and reactions of ω-CF3O-substituted aliphatic sulfonyl chlorides. Journal of Fluorine Chemistry 2021;246:109799. [DOI: 10.1016/j.jfluchem.2021.109799] [Reference Citation Analysis]
36 Doobary S, Poole DL, Lennox AJJ. Intramolecular Alkene Fluoroarylation of Phenolic Ethers Enabled by Electrochemically Generated Iodane. J Org Chem 2021;86:16095-103. [PMID: 34766770 DOI: 10.1021/acs.joc.1c01946] [Reference Citation Analysis]
37 Pothireddy M, Bhukta S, Babu PV, Thirupathi B, Dandela R. Synthetic method to access fluorinated 2-benzylpyridines by using Negishi coupling reaction. Synthetic Communications. [DOI: 10.1080/00397911.2022.2037651] [Reference Citation Analysis]
38 Maria Faisca Phillips A, Pombeiro AJL. Recent Developments in Enantioselective Organocatalytic Cascade Reactions for the Construction of Halogenated Ring Systems. Eur J Org Chem 2021;2021:3938-69. [DOI: 10.1002/ejoc.202100364] [Cited by in Crossref: 2] [Cited by in F6Publishing: 1] [Article Influence: 2.0] [Reference Citation Analysis]
39 Yang J, Ponra S, Li X, Peters BBC, Massaro L, Zhou T, Andersson PG. Catalytic enantioselective synthesis of fluoromethylated stereocenters by asymmetric hydrogenation. Chem Sci 2022;13:8590-6. [DOI: 10.1039/d2sc02685f] [Reference Citation Analysis]
40 Uno H, Fujimoto D, Harada K, Tanaka C, Shibata N. Synthesis of Tetra-Substituted Trifluoromethyl-3,1-Benzoxazines by Transition-Metal-Catalyzed Decarboxylative Cyclization of N-Benzoyl Benzoxazinones. ChemistryOpen 2021;10:518-22. [PMID: 33605087 DOI: 10.1002/open.202000360] [Cited by in Crossref: 1] [Cited by in F6Publishing: 1] [Article Influence: 1.0] [Reference Citation Analysis]
41 Shcherbakov KV, Panova MA, Burgart YV, Zarubaev VV, Gerasimova NA, Evstigneeva NP, Saloutin VI. The synthesis and biological evaluation of A- and B-ring fluorinated flavones and their key intermediates. Journal of Fluorine Chemistry 2021;249:109857. [DOI: 10.1016/j.jfluchem.2021.109857] [Reference Citation Analysis]
42 Tanács D, Berkecz R, Shahmohammadi S, Forró E, Armstrong DW, Péter A, Ilisz I. Macrocyclic glycopeptides- and derivatized cyclofructan-based chiral stationary phases for the enantioseparation of fluorinated ß-phenylalanine analogs. Journal of Pharmaceutical and Biomedical Analysis 2022;219:114912. [DOI: 10.1016/j.jpba.2022.114912] [Reference Citation Analysis]
43 Fu J, Tsapy Takia IR, Chen P, Liu W, Jiang C, Yao W, Zeng X, Wang Y, Han X. Synthesis of 2-chromanone-fused [3.2.0] bicycles through a phosphine-mediated tandem [3 + 2] cyclization/intramolecular Wittig reaction. Org Chem Front 2021;8:6323-9. [DOI: 10.1039/d1qo01013a] [Reference Citation Analysis]
44 Han J, Kiss L, Mei H, Remete AM, Ponikvar-Svet M, Sedgwick DM, Roman R, Fustero S, Moriwaki H, Soloshonok VA. Chemical Aspects of Human and Environmental Overload with Fluorine. Chem Rev 2021;121:4678-742. [PMID: 33723999 DOI: 10.1021/acs.chemrev.0c01263] [Cited by in Crossref: 11] [Cited by in F6Publishing: 1] [Article Influence: 11.0] [Reference Citation Analysis]
45 Schäfer M, Stünkel T, Daniliuc CG, Gilmour R. Regio- and Enantioselective Intermolecular Aminofluorination of Alkenes via Iodine(I)/Iodine(III) Catalysis. Angew Chem Int Ed Engl 2022;61:e202205508. [PMID: 35583965 DOI: 10.1002/anie.202205508] [Cited by in Crossref: 1] [Cited by in F6Publishing: 1] [Article Influence: 1.0] [Reference Citation Analysis]
46 Liu A, Han J, Nakano A, Konno H, Moriwaki H, Abe H, Izawa K, Soloshonok VA. New pharmaceuticals approved by FDA in 2020: Small-molecule drugs derived from amino acids and related compounds. Chirality 2022;34:86-103. [PMID: 34713503 DOI: 10.1002/chir.23376] [Reference Citation Analysis]
47 Grollier K, Chefdeville E, Jeanneau E, Billard T. Aromatic Trifluoromethylselenolation via Pd-catalyzed C-H functionalization. Chemistry 2021;27:12910-6. [PMID: 34142744 DOI: 10.1002/chem.202102121] [Cited by in Crossref: 1] [Article Influence: 1.0] [Reference Citation Analysis]
48 Kawai K, Uno H, Fujimoto D, Shibata N. Transition‐Metal Free Catalytic Synthesis of Trifluoromethyl Indolines by [4+1] Cycloaddition of Trifluoromethyl Benzoxazinones with Sulfur Ylides. Helv Chim Acta 2021;104. [DOI: 10.1002/hlca.202000217] [Cited by in Crossref: 2] [Cited by in F6Publishing: 1] [Article Influence: 2.0] [Reference Citation Analysis]
49 Levin VV, Dilman AD. One-pot synthesis of α-trifluoromethylstyrenes from aryl ketones and the Ruppert–Prakash reagent. Mendeleev Communications 2021;31:684-5. [DOI: 10.1016/j.mencom.2021.09.030] [Cited by in Crossref: 2] [Cited by in F6Publishing: 2] [Article Influence: 2.0] [Reference Citation Analysis]
50 Ma Y, Lv L, Li Z. β-Perfluoroalkyl Peroxides as Fluorinated C3-Building Blocks for the Construction of Benzo[4,5]imidazo[1,2-a]pyridines. J Org Chem 2022;87:1564-73. [PMID: 34989560 DOI: 10.1021/acs.joc.1c02589] [Reference Citation Analysis]
51 Zanakhov TO, Galenko EE, Novikov MS, Khlebnikov AF. An isoxazole strategy for the synthesis of 4-oxo-1,4-dihydropyridine-3-carboxylates. Beilstein J Org Chem 2022;18:738-45. [DOI: 10.3762/bjoc.18.74] [Reference Citation Analysis]
52 Liu J, Xiang H, Jiang L, Yi W. Chemoselective desulfurization-fluorination/bromination of carbonofluoridothioates for the O-trifluoromethylation and O-bromodifluoromethylation of alcohols. Sci China Chem 2021;64:1372-9. [DOI: 10.1007/s11426-021-1028-6] [Cited by in Crossref: 2] [Cited by in F6Publishing: 1] [Article Influence: 2.0] [Reference Citation Analysis]
53 Xia P, Liu F, Li S, Xiao J. Tunable photocatalytic oxysulfonylation and chlorosulfonylation of α-CF 3 alkenes with sulfonyl chlorides. Org Chem Front 2022;9:709-14. [DOI: 10.1039/d1qo01686e] [Cited by in Crossref: 2] [Cited by in F6Publishing: 2] [Article Influence: 2.0] [Reference Citation Analysis]
54 Glyn RJ, Pattison G. Effects of Replacing Oxygenated Functionality with Fluorine on Lipophilicity. J Med Chem 2021;64:10246-59. [PMID: 34213355 DOI: 10.1021/acs.jmedchem.1c00668] [Reference Citation Analysis]
55 Elkina NA, Shchegolkov EV, Burgart YV, Agafonova NA, Perminova AN, Gerasimova NA, Makhaeva GF, Rudakova EV, Kovaleva NV, Boltneva NP, Serebryakova OG, Borisevich SS, Evstigneeva NP, Zilberberg NV, Kungurov NV, Saloutin VI. Synthesis and biological evaluation of polyfluoroalkyl-containing 4-arylhydrazinylidene-isoxazoles as antifungal agents with antioxidant activity. Journal of Fluorine Chemistry 2022;254:109935. [DOI: 10.1016/j.jfluchem.2021.109935] [Reference Citation Analysis]
56 Znidar D, Dallinger D, Kappe CO. Practical Guidelines for the Safe Use of Fluorine Gas Employing Continuous Flow Technology. ACS Chem Health Saf . [DOI: 10.1021/acs.chas.1c00097] [Cited by in Crossref: 2] [Cited by in F6Publishing: 1] [Article Influence: 2.0] [Reference Citation Analysis]
57 Shevchuk M, Wang Q, Pajkert R, Xu J, Mei H, Röschenthaler G, Han J. Recent Advances in Synthesis of Difluoromethylene Phosphonates for Biological Applications. Adv Synth Catal 2021;363:2912-68. [DOI: 10.1002/adsc.202001464] [Cited by in Crossref: 5] [Cited by in F6Publishing: 1] [Article Influence: 5.0] [Reference Citation Analysis]
58 Supranovich VI, Volodin AD, Korlyukov AA, Hu J, Dilman AD. Reaction of (bromodifluoromethyl)trimethylsilane with HMPA: Structural studies. Journal of Fluorine Chemistry 2021;250:109881. [DOI: 10.1016/j.jfluchem.2021.109881] [Reference Citation Analysis]
59 Liu J, Lin W, Sorochinsky AE, Butler G, Landa A, Han J, Soloshonok VA. Successful trifluoromethoxy-containing pharmaceuticals and agrochemicals. Journal of Fluorine Chemistry 2022. [DOI: 10.1016/j.jfluchem.2022.109978] [Reference Citation Analysis]
60 Logvinenko IG, Kondratov IS, Pridma SO, Tolmachova NA, Morev RN, Dolovanyuk VG, Boretskyi AL, Stepanyuk RO, Trofimchuk SA, Mück-lichtenfeld C, Daniliuc CG, Haufe G. Synthesis and physical chemical properties of CF3O-containg secondary amines – perspective building blocks for Drug Discovery. Journal of Fluorine Chemistry 2022. [DOI: 10.1016/j.jfluchem.2022.109990] [Reference Citation Analysis]