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Sun Z, Xiao L, Chen Y, Wang J, Zeng F, Zhang H, Zhang J, Yang K, Hu YJ. Constructive On-DNA Abramov Reaction and Pudovik Reaction for DEL Synthesis. ACS Med Chem Lett 2023. [DOI: 10.1021/acsmedchemlett.3c00022] [Reference Citation Analysis]
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Luo A, Zhou H, Hua Q, An Y, Ma H, Zhao X, Yang K, Hu YJ. Development of the Inverse Sonogashira Reaction for DEL Synthesis. ACS Med Chem Lett 2023;14:270-7. [PMID: 36923912 DOI: 10.1021/acsmedchemlett.2c00477] [Cited by in Crossref: 1] [Article Influence: 1.0] [Reference Citation Analysis]
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Fang X, Liao H, Fan X, Wang Y, Wang H, Zhang G, Fang W, Li Y, Li Y. Incorporation of viridicatin alkaloid-like scaffolds into DNA-encoded chemical libraries. Org Biomol Chem 2023;21:2162-6. [PMID: 36799438 DOI: 10.1039/d2ob02278h] [Reference Citation Analysis]
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Stanway-Gordon HA, Odger JA, Waring MJ. Development of a Micellar-Promoted Heck Reaction for the Synthesis of DNA-Encoded Libraries. Bioconjug Chem 2023. [PMID: 36883323 DOI: 10.1021/acs.bioconjchem.3c00051] [Reference Citation Analysis]
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Li L, Matsuo B, Levitre G, McClain EJ, Voight EA, Crane EA, Molander GA. Dearomative intermolecular [2 + 2] photocycloaddition for construction of C(sp(3))-rich heterospirocycles on-DNA. Chem Sci 2023;14:2713-20. [PMID: 36908969 DOI: 10.1039/d3sc00144j] [Reference Citation Analysis]
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Krishna Sunkari Y, Kumar Siripuram V, Flajolet M. Diversity-Oriented Synthesis (DOS) of On-DNA Peptidomimetics from Acid-Derived Phosphonium Ylides. Chemistry 2023;29:e202203037. [PMID: 36653313 DOI: 10.1002/chem.202203037] [Reference Citation Analysis]
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Wen X, Wu X, Jin R, Lu X. Privileged heterocycles for DNA-encoded library design and hit-to-lead optimization. Eur J Med Chem 2023;248:115079. [PMID: 36669370 DOI: 10.1016/j.ejmech.2022.115079] [Reference Citation Analysis]
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Mahdavi-Amiri Y, Hu MSJ, Frias N, Movahedi M, Csakai A, Marcaurelle LA, Hili R. Photoredox-catalysed hydroaminoalkylation of on-DNA N-arylamines. Org Biomol Chem 2023;21:1463-7. [PMID: 36655521 DOI: 10.1039/d2ob01956f] [Reference Citation Analysis]
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Matsuo B, Granados A, Levitre G, Molander GA. Photochemical Methods Applied to DNA Encoded Library (DEL) Synthesis. Acc Chem Res 2023;56:385-401. [PMID: 36656960 DOI: 10.1021/acs.accounts.2c00778] [Reference Citation Analysis]
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Montoya AL, Glavatskikh M, Halverson BJ, Yuen LH, Schüler H, Kireev D, Franzini RM. Combining pharmacophore models derived from DNA-encoded chemical libraries with structure-based exploration to predict Tankyrase 1 inhibitors. Eur J Med Chem 2023;246:114980. [PMID: 36495630 DOI: 10.1016/j.ejmech.2022.114980] [Reference Citation Analysis]
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Chheda PR, Simmons N, Schuman DP, Shi Z. Photoredox-Mediated Deoxygenative Alkylation of DNA-Tagged Alkenes with Activated Alcohols. Org Lett 2022;24:9514-9. [PMID: 36541781 DOI: 10.1021/acs.orglett.2c03994] [Reference Citation Analysis]
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Luo A, Zhou H, Zhou Q, Hua Q, Zhao X, Yu X, Yang K, Hu YJ. On-DNA Alkyne Iodination and Acetylenic Coupling as a Useful Tool for DEL Synthesis. Bioconjug Chem 2022;33:2299-306. [PMID: 36450158 DOI: 10.1021/acs.bioconjchem.2c00471] [Reference Citation Analysis]
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Young RJ, Flitsch SL, Grigalunas M, Leeson PD, Quinn RJ, Turner NJ, Waldmann H. The Time and Place for Nature in Drug Discovery. JACS Au 2022;2:2400-2416. [DOI: 10.1021/jacsau.2c00415] [Reference Citation Analysis]
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Janin YL. On drug discovery against infectious diseases and academic medicinal chemistry contributions. Beilstein J Org Chem 2022;18:1355-78. [DOI: 10.3762/bjoc.18.141] [Reference Citation Analysis]
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Yen-Pon E, Li L, Levitre G, Majhi J, McClain EJ, Voight EA, Crane EA, Molander GA. On-DNA Hydroalkylation to Introduce Diverse Bicyclo[1.1.1]pentanes and Abundant Alkyls via Halogen Atom Transfer. J Am Chem Soc 2022;144:12184-91. [PMID: 35759692 DOI: 10.1021/jacs.2c03025] [Cited by in Crossref: 5] [Cited by in F6Publishing: 4] [Article Influence: 5.0] [Reference Citation Analysis]
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Chheda PR, Simmons N, Schuman DP, Shi Z. Palladium-Mediated Carbonylative Suzuki Coupling for DNA-Encoded Library Synthesis. Org Lett 2022. [PMID: 35830624 DOI: 10.1021/acs.orglett.2c02113] [Cited by in F6Publishing: 1] [Reference Citation Analysis]
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Eom S, Kwon T, Lee DY, Park CH, Kim HJ. Copper-Mediated Three-Component Reaction for the Synthesis of N-Acylsulfonamide on DNA. Org Lett 2022. [PMID: 35775977 DOI: 10.1021/acs.orglett.2c01675] [Reference Citation Analysis]
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Sun J, Nie Q, Fang X, He Z, Zhang G, Li Y, Li Y. Vinyl azide as a synthon for DNA-compatible divergent transformations into N-heterocycles. Org Biomol Chem 2022;20:5045-9. [PMID: 35703385 DOI: 10.1039/d2ob00862a] [Cited by in Crossref: 1] [Cited by in F6Publishing: 2] [Article Influence: 1.0] [Reference Citation Analysis]
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Chheda PR, Simmons N, Schuman DP, Shi Z. Palladium-Mediated C–N Coupling of DNA-Conjugated (Hetero)aryl Halides with Aliphatic and (Hetero)aromatic Amines. Org Lett . [DOI: 10.1021/acs.orglett.2c01175] [Cited by in Crossref: 2] [Cited by in F6Publishing: 3] [Article Influence: 2.0] [Reference Citation Analysis]
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Cai K, Ran Y, Sun W, Gao S, Li J, Wan J, Liu G. Palladium-Mediated Hydroamination of DNA-Conjugated Aryl Alkenes. Front Chem 2022;10:851674. [DOI: 10.3389/fchem.2022.851674] [Reference Citation Analysis]
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Adamik R, Buchholcz B, Darvas F, Sipos G, Novák Z. The Potential of Micellar Media in the Synthesis of DNA-Encoded Libraries. Chemistry 2022;28:e202103967. [PMID: 35019168 DOI: 10.1002/chem.202103967] [Cited by in Crossref: 1] [Cited by in F6Publishing: 2] [Article Influence: 1.0] [Reference Citation Analysis]
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Gui Y, Wong CS, Zhao G, Xie C, Hou R, Li Y, Li G, Li X. Converting Double-Stranded DNA-Encoded Libraries (DELs) to Single-Stranded Libraries for More Versatile Selections. ACS Omega 2022;7:11491-500. [PMID: 35415338 DOI: 10.1021/acsomega.2c01152] [Cited by in Crossref: 3] [Cited by in F6Publishing: 3] [Article Influence: 3.0] [Reference Citation Analysis]
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Sun ZM, Yang SG, Xue LJ, Zhang J, Yang K, Hu YJ. N-Alkyl Linkers for DNA-Encoded Chemical Libraries. Chem Asian J 2022;:e202200016. [PMID: 35254005 DOI: 10.1002/asia.202200016] [Cited by in Crossref: 1] [Cited by in F6Publishing: 1] [Article Influence: 1.0] [Reference Citation Analysis]
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Yang S, Zhao G, Gao Y, Sun Y, Zhang G, Fan X, Li Y, Li Y. In-solution direct oxidative coupling for the integration of sulfur/selenium into DNA-encoded chemical libraries. Chem Sci 2022;13:2604-13. [PMID: 35340849 DOI: 10.1039/d1sc06268a] [Cited by in Crossref: 10] [Cited by in F6Publishing: 10] [Article Influence: 10.0] [Reference Citation Analysis]
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Anderson MJ, Castan IFSF, Graham JS, Hassan H, Odger J, Salvini CLA, Taylor C, Waring MJ. Advancements in DEL-Compatible Chemical Reactions. Topics in Medicinal Chemistry 2022. [DOI: 10.1007/7355_2022_151] [Reference Citation Analysis]
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Chines S, Ehrt C, Potowski M, Biesenkamp F, Grützbach L, Brunner S, van den Broek F, Bali S, Ickstadt K, Brunschweiger A. Navigating chemical reaction space – application to DNA-encoded chemistry. Chem Sci 2022;13:11221-31. [DOI: 10.1039/d2sc02474h] [Reference Citation Analysis]
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Morgan BA. A Perspective on 30 Years of DNA-Encoded Chemistry. Topics in Medicinal Chemistry 2022. [DOI: 10.1007/7355_2022_152] [Reference Citation Analysis]
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Zhang Y, Franzini RM. Design Considerations in Constructing and Screening DNA-Encoded Libraries. Topics in Medicinal Chemistry 2022. [DOI: 10.1007/7355_2022_147] [Reference Citation Analysis]
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Gao Y, Zhao G, He P, Zhang G, Li Y, Li Y. DNA-Compatible Synthesis of α,β-Epoxyketones for DNA-Encoded Chemical Libraries. Bioconjug Chem 2021. [PMID: 34927428 DOI: 10.1021/acs.bioconjchem.1c00567] [Cited by in Crossref: 7] [Cited by in F6Publishing: 7] [Article Influence: 3.5] [Reference Citation Analysis]
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