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For: Grygorenko OO, Volochnyuk DM, Ryabukhin SV, Judd DB. The Symbiotic Relationship Between Drug Discovery and Organic Chemistry. Chemistry 2020;26:1196-237. [PMID: 31429510 DOI: 10.1002/chem.201903232] [Cited by in Crossref: 43] [Cited by in F6Publishing: 19] [Article Influence: 14.3] [Reference Citation Analysis]
Number Citing Articles
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2 Li S, Pissarnitski D, Nowak T, Wleklinski M, Krska SW. Merging Late-Stage Diversification with Solid-Phase Peptide Synthesis Enabled by High-Throughput On-Resin Reaction Screening. ACS Catal 2022;12:3201-10. [DOI: 10.1021/acscatal.1c05502] [Reference Citation Analysis]
3 Omelian TV, Dobrydnev AV, Utchenko OY, Ostapchuk EN, Konovalova IS, Volovenko YM. The reactivity of tetrahydropyrrolo[1,2-b]isothiazol-3(2H)-one 1,1-dioxides. Monatsh Chem 2020;151:1759-72. [DOI: 10.1007/s00706-020-02694-3] [Cited by in Crossref: 4] [Article Influence: 2.0] [Reference Citation Analysis]
4 Sotnik SO, Subota AI, Kliuchynskyi AY, Yehorov DV, Lytvynenko AS, Rozhenko AB, Kolotilov SV, Ryabukhin SV, Volochnyuk DM. Cu-Catalyzed Pyridine Synthesis via Oxidative Annulation of Cyclic Ketones with Propargylamine. J Org Chem 2021;86:7315-25. [PMID: 33977713 DOI: 10.1021/acs.joc.0c03038] [Reference Citation Analysis]
5 Zabolotna Y, Lin A, Horvath D, Marcou G, Volochnyuk DM, Varnek A. Chemography: Searching for Hidden Treasures. J Chem Inf Model 2021;61:179-88. [PMID: 33334102 DOI: 10.1021/acs.jcim.0c00936] [Cited by in Crossref: 3] [Cited by in F6Publishing: 3] [Article Influence: 1.5] [Reference Citation Analysis]
6 Kyrylchuk A, Kravets I, Cherednichenko A, Tararina V, Kapeliukha A, Dudenko D, Protopopov M. Creation of targeted compound libraries based on 3D shape recognition. Mol Divers 2022. [PMID: 35608807 DOI: 10.1007/s11030-022-10447-z] [Reference Citation Analysis]
7 Bozhanov VI, Bohdan DP, Borysov OV, Silin AV, Zaremba OV, Avramenko MM, Volochnyuk DM, Ryabukhin SV, Gavrilenko KS. Straightforward Synthesis of Functionalized 4,5,6,7‐Tetrahydro‐pyrazolo[1,5‐a]pyrazines – Important Building Blocks for Medicinal Chemistry. ChemistrySelect 2022;7. [DOI: 10.1002/slct.202104287] [Reference Citation Analysis]
8 Yue C, Gu L. Understanding and Learning of Ionic Organic Reactions in Organic Chemistry Based on Acid–Base Theory. J Chem Educ . [DOI: 10.1021/acs.jchemed.1c01130] [Reference Citation Analysis]
9 Chessari G, Grainger R, Holvey RS, Ludlow RF, Mortenson PN, Rees DC. C-H functionalisation tolerant to polar groups could transform fragment-based drug discovery (FBDD). Chem Sci 2021;12:11976-85. [PMID: 34667563 DOI: 10.1039/d1sc03563k] [Cited by in Crossref: 1] [Article Influence: 1.0] [Reference Citation Analysis]
10 Kokhan SO, Valter YB, Tymtsunik AV, Komarov IV, Grygorenko OO. 3-Carboxy-/3-Aminobicyclo[1.1.1]pentane-Derived Sulfonamides and Sulfonyl Fluorides - Advanced Bifunctional Reagents for Organic Synthesis and Drug Discovery: 3-Carboxy-/3-Aminobicyclo[1.1.1]pentane-Derived Sulfonamides and Sulfonyl Fluorides - Advanced Bifunctional Reagents for Organic Synthesis and Drug Di. Eur J Org Chem 2020;2020:2210-6. [DOI: 10.1002/ejoc.202000303] [Cited by in Crossref: 6] [Cited by in F6Publishing: 2] [Article Influence: 3.0] [Reference Citation Analysis]
11 Stepannikova KO, Vashchenko BV, Grygorenko OO, Gorichko MV, Cherepakha AY, Moroz YS, Volovenko YM, Zhersh S. Synthesis of Spirocyclic β- and γ-Sultams by One-Pot Reductive Cyclization of Cyanoalkylsulfonyl Fluorides: Synthesis of Spirocyclic β- and γ-Sultams by One-Pot Reductive Cyclization of Cyanoalkylsulfonyl Fluorides. Eur J Org Chem . [DOI: 10.1002/ejoc.202000351] [Cited by in Crossref: 4] [Cited by in F6Publishing: 1] [Article Influence: 2.0] [Reference Citation Analysis]
12 Wang T, Kadow JF, Meanwell NA. Innovation in the discovery of the HIV-1 attachment inhibitor temsavir and its phosphonooxymethyl prodrug fostemsavir. Med Chem Res 2021;:1-26. [PMID: 34602806 DOI: 10.1007/s00044-021-02787-6] [Reference Citation Analysis]
13 Schütz C, Hodzic A, Hamed M, Abdelsamie AS, Kany AM, Bauer M, Röhrig T, Schmelz S, Scrima A, Blankenfeldt W, Empting M. Divergent synthesis and biological evaluation of 2-(trifluoromethyl)pyridines as virulence-attenuating inverse agonists targeting PqsR. Eur J Med Chem 2021;226:113797. [PMID: 34520957 DOI: 10.1016/j.ejmech.2021.113797] [Reference Citation Analysis]
14 Grygorenko OO, Hryshchuk OV. Cyclopropylation of heterocyclic cores using cyclopropylboronic derivatives (microreview). Chem Heterocycl Comp 2020;56:39-41. [DOI: 10.1007/s10593-020-02619-2] [Cited by in Crossref: 6] [Article Influence: 3.0] [Reference Citation Analysis]
15 Saldívar-González FI, Medina-Franco JL. Approaches for enhancing the analysis of chemical space for drug discovery. Expert Opin Drug Discov 2022. [PMID: 35640229 DOI: 10.1080/17460441.2022.2084608] [Reference Citation Analysis]
16 Ghosh C, Patra D, Bala N, Majumder I, Sepay N, Mukhopadhyay P, Das S, Kundu R, Drew MGB, León AR, Ghosh T, Pradhan M. A family of amphiphilic dioxidovanadium(V) hydrazone complexes as potent carbonic anhydrase inhibitors along with anti-diabetic and cytotoxic activities. Biometals 2022. [PMID: 35355153 DOI: 10.1007/s10534-022-00384-7] [Reference Citation Analysis]
17 Kleban I, Radchenko DS, Tymtsunik AV, Shuvakin S, Konovets AI, Rassukana Y, Grygorenko OO. Cyclopropyl boronic derivatives in parallel synthesis of sp3-enriched compound libraries. Monatsh Chem 2020;151:953-62. [DOI: 10.1007/s00706-020-02619-0] [Cited by in Crossref: 2] [Cited by in F6Publishing: 1] [Article Influence: 1.0] [Reference Citation Analysis]
18 St Denis JD, Hall RJ, Murray CW, Heightman TD, Rees DC. Fragment-based drug discovery: opportunities for organic synthesis. RSC Med Chem 2020;12:321-9. [PMID: 34041484 DOI: 10.1039/d0md00375a] [Cited by in Crossref: 6] [Cited by in F6Publishing: 1] [Article Influence: 3.0] [Reference Citation Analysis]
19 Weis E, Johansson M, Korsgren P, Martín-matute B, Johansson MJ. Merging Directed C–H Activations with High-Throughput Experimentation: Development of Iridium-Catalyzed C–H Aminations Applicable to Late-Stage Functionalization. JACS Au. [DOI: 10.1021/jacsau.2c00039] [Reference Citation Analysis]
20 Cui Y. Landscaping Agricultural and Animal Husbandry Production Park Using Lightweight Deep Reinforcement Learning under Circular Symbiosis Concept. Comput Intell Neurosci 2022;2022:8410996. [PMID: 35694577 DOI: 10.1155/2022/8410996] [Reference Citation Analysis]
21 Nakamura T, Sakaue S, Fujii K, Harabuchi Y, Maeda S, Iwata S. Selecting molecules with diverse structures and properties by maximizing submodular functions of descriptors learned with graph neural networks. Sci Rep 2022;12:1124. [PMID: 35064170 DOI: 10.1038/s41598-022-04967-9] [Reference Citation Analysis]
22 Grygorenko OO, Vashchenko BV, Blahun OP, Zhersh S. Saturated Bicyclic Sultams. Eur J Org Chem 2020;2020:5787-800. [DOI: 10.1002/ejoc.202000603] [Cited by in Crossref: 5] [Cited by in F6Publishing: 1] [Article Influence: 2.5] [Reference Citation Analysis]
23 Chamakuri S, Lu S, Ucisik MN, Bohren KM, Chen YC, Du HC, Faver JC, Jimmidi R, Li F, Li JY, Nyshadham P, Palmer SS, Pollet J, Qin X, Ronca SE, Sankaran B, Sharma KL, Tan Z, Versteeg L, Yu Z, Matzuk MM, Palzkill T, Young DW. DNA-encoded chemistry technology yields expedient access to SARS-CoV-2 Mpro inhibitors. Proc Natl Acad Sci U S A 2021;118:e2111172118. [PMID: 34426525 DOI: 10.1073/pnas.2111172118] [Reference Citation Analysis]
24 Grygorenko OO, Moskvina VS, Kleban I, Hryshchyk OV. Synthesis of saturated and partially saturated heterocyclic boronic derivatives. Tetrahedron 2022;104:132605. [DOI: 10.1016/j.tet.2021.132605] [Cited by in Crossref: 1] [Cited by in F6Publishing: 1] [Article Influence: 1.0] [Reference Citation Analysis]
25 Kleban I, Krokhmaliuk Y, Reut S, Shuvakin S, Pendyukh VV, Khyzhan OI, Yarmoliuk DS, Tymtsunik AV, Rassukana YV, Grygorenko OO. Multigram Synthesis of Heterabicyclo[n.1.0]alkan‐1‐yl Trifluoroborates. European J Organic Chem 2021;2021:6551-60. [DOI: 10.1002/ejoc.202000977] [Cited by in Crossref: 2] [Cited by in F6Publishing: 1] [Article Influence: 1.0] [Reference Citation Analysis]
26 Demchuk OP, Hryshchuk OV, Vashchenko BV, Kozytskiy AV, Tymtsunik AV, Komarov IV, Grygorenko OO. Photochemical [2 + 2] Cycloaddition of Alkenyl Boronic Derivatives: An Entry into 3-Azabicyclo[3.2.0]heptane Scaffold. J Org Chem 2020;85:5927-40. [PMID: 32233365 DOI: 10.1021/acs.joc.0c00265] [Cited by in Crossref: 5] [Cited by in F6Publishing: 3] [Article Influence: 2.5] [Reference Citation Analysis]
27 Chalyk BA, Khutorianskyi A, Lysenko A, Fil Y, Kuchkovska YO, Gavrilenko KS, Bakanovych I, Moroz YS, Gorlova AO, Grygorenko OO. Regioselective Synthesis of Functionalized 3- or 5-Fluoroalkyl Isoxazoles and Pyrazoles from Fluoroalkyl Ynones and Binucleophiles. J Org Chem 2019;84:15212-25. [PMID: 31661620 DOI: 10.1021/acs.joc.9b02258] [Cited by in Crossref: 9] [Cited by in F6Publishing: 4] [Article Influence: 3.0] [Reference Citation Analysis]
28 Biletskyi B, Colonna P, Masson K, Parrain JL, Commeiras L, Chouraqui G. Small rings in the bigger picture: ring expansion of three- and four-membered rings to access larger all-carbon cyclic systems. Chem Soc Rev 2021;50:7513-38. [PMID: 34002179 DOI: 10.1039/d0cs01396j] [Cited by in Crossref: 5] [Cited by in F6Publishing: 1] [Article Influence: 5.0] [Reference Citation Analysis]
29 Logvinenko IG, Kondratov IS, Dobrydnev AV, Kozytskiy AV, Grygorenko OO. Synthesis and reactions of ω-CF3O-substituted aliphatic sulfonyl chlorides. Journal of Fluorine Chemistry 2021;246:109799. [DOI: 10.1016/j.jfluchem.2021.109799] [Reference Citation Analysis]
30 Guariento S, Biagetti M, Ronchi P. Non-regioselective functionalization: an underestimate chemical diversity generator in medicinal chemistry. Future Med Chem 2021;13:595-9. [PMID: 33657835 DOI: 10.4155/fmc-2021-0011] [Reference Citation Analysis]
31 Chernykh AV, Chernykh AV, Radchenko DS, Chheda PR, Rusanov EB, Grygorenko OO, Spies MA, Volochnyuk DM, Komarov IV. A stereochemical journey around spirocyclic glutamic acid analogs. Org Biomol Chem 2022;20:3183-200. [PMID: 35348173 DOI: 10.1039/d2ob00146b] [Reference Citation Analysis]
32 Serafim MSM, Dos Santos Júnior VS, Gertrudes JC, Maltarollo VG, Honorio KM. Machine learning techniques applied to the drug design and discovery of new antivirals: a brief look over the past decade. Expert Opin Drug Discov 2021;16:961-75. [PMID: 33957833 DOI: 10.1080/17460441.2021.1918098] [Cited by in Crossref: 1] [Cited by in F6Publishing: 1] [Article Influence: 1.0] [Reference Citation Analysis]
33 Mittersteiner M, Bonacorso HG, Martins MAP, Zanatta N. Haloacetylated Enol Ethers: a Way Out for the Regioselective Synthesis of Biologically Active Heterocycles. Eur J Org Chem 2021;2021:3886-911. [DOI: 10.1002/ejoc.202100495] [Cited by in Crossref: 5] [Cited by in F6Publishing: 4] [Article Influence: 5.0] [Reference Citation Analysis]
34 Gomez-angel AR, Donald JR, Firth JD, De Fusco C, Ian Storer R, Cox DJ, O’brien P. Synthesis and functionalisation of a bifunctional normorphan 3D building block for medicinal chemistry. Tetrahedron 2021;83:131961. [DOI: 10.1016/j.tet.2021.131961] [Cited by in Crossref: 3] [Cited by in F6Publishing: 1] [Article Influence: 3.0] [Reference Citation Analysis]
35 Grygorenko OO, Radchenko DS, Dziuba I, Chuprina A, Gubina KE, Moroz YS. Generating Multibillion Chemical Space of Readily Accessible Screening Compounds. iScience 2020;23:101681. [DOI: 10.1016/j.isci.2020.101681] [Cited by in Crossref: 14] [Cited by in F6Publishing: 9] [Article Influence: 7.0] [Reference Citation Analysis]
36 Ramsden JI, Cosgrove SC, Turner NJ. Is it time for biocatalysis in fragment-based drug discovery? Chem Sci 2020;11:11104-12. [PMID: 34094353 DOI: 10.1039/d0sc04103c] [Cited by in Crossref: 5] [Cited by in F6Publishing: 1] [Article Influence: 2.5] [Reference Citation Analysis]
37 Ronzon Q, Zhang W, Casaretto N, Mouray E, Florent I, Nay B. Programmed Multiple C-H Bond Functionalization of the Privileged 4-hydroxyquinoline Template. Chemistry 2021;27:7764-72. [PMID: 33848033 DOI: 10.1002/chem.202100929] [Reference Citation Analysis]
38 Zabolotna Y, Volochnyuk DM, Ryabukhin SV, Horvath D, Gavrilenko KS, Marcou G, Moroz YS, Oksiuta O, Varnek A. A Close-up Look at the Chemical Space of Commercially Available Building Blocks for Medicinal Chemistry. J Chem Inf Model 2021. [PMID: 34928600 DOI: 10.1021/acs.jcim.1c00811] [Reference Citation Analysis]
39 Aguilar-Morales CM, Araujo-Huitrado JG, López-Hernández Y, Contreras-Celedón C, Islas-Jácome A, Granados-López AJ, Solorio-Alvarado CR, López JA, Chacón-García L, Cortés-García CJ. A One-Pot Six-Component Reaction for the Synthesis of 1,5-Disubstituted Tetrazol-1,2,3-Triazole Hybrids and Their Cytotoxic Activity against the MCF-7 Cell Line. Molecules 2021;26:6104. [PMID: 34684686 DOI: 10.3390/molecules26206104] [Reference Citation Analysis]
40 Grigalunas M, Brakmann S, Waldmann H. Chemical Evolution of Natural Product Structure. J Am Chem Soc . [DOI: 10.1021/jacs.1c11270] [Cited by in Crossref: 2] [Cited by in F6Publishing: 1] [Article Influence: 2.0] [Reference Citation Analysis]
41 Oderinde MS, Jin S, Dhar TM, Meanwell NA, Mathur A, Kempson J. Advances in the synthesis of three-dimensional molecular architectures by dearomatizing photocycloadditions. Tetrahedron 2022;103:132087. [DOI: 10.1016/j.tet.2021.132087] [Cited by in Crossref: 2] [Cited by in F6Publishing: 2] [Article Influence: 2.0] [Reference Citation Analysis]
42 Vaškevičius M, Kapočiūtė-Dzikienė J, Šlepikas L. Prediction of Chromatography Conditions for Purification in Organic Synthesis Using Deep Learning. Molecules 2021;26:2474. [PMID: 33922736 DOI: 10.3390/molecules26092474] [Reference Citation Analysis]
43 Laird TS, Flores N, Leveau JHJ. Bacterial catabolism of indole-3-acetic acid. Appl Microbiol Biotechnol 2020;104:9535-50. [PMID: 33037916 DOI: 10.1007/s00253-020-10938-9] [Cited by in Crossref: 3] [Cited by in F6Publishing: 2] [Article Influence: 1.5] [Reference Citation Analysis]
44 Pennington LD, Aquila BM, Choi Y, Valiulin RA, Muegge I. Positional Analogue Scanning: An Effective Strategy for Multiparameter Optimization in Drug Design. J Med Chem 2020;63:8956-76. [PMID: 32330036 DOI: 10.1021/acs.jmedchem.9b02092] [Cited by in Crossref: 9] [Cited by in F6Publishing: 7] [Article Influence: 4.5] [Reference Citation Analysis]
45 Vaskevych AI, Savinchuk NO, Vaskevych RI, Rusanov EB, Grygorenko OO, Vovk MV. The PIFA-initiated oxidative cyclization of 2-(3-butenyl)quinazolin-4(3H)-ones - an efficient approach to 1-(hydroxymethyl)-2,3-dihydropyrrolo[1,2-a]quinazolin-5(1H)-ones. Beilstein J Org Chem 2021;17:2787-94. [PMID: 34900009 DOI: 10.3762/bjoc.17.189] [Reference Citation Analysis]
46 Grygorenko OO, Volochnyuk DM, Vashchenko BV. Emerging Building Blocks for Medicinal Chemistry: Recent Synthetic Advances. European J Organic Chem 2021;2021:6478-510. [DOI: 10.1002/ejoc.202100857] [Cited by in Crossref: 1] [Article Influence: 1.0] [Reference Citation Analysis]
47 Andriashvili VA, Zhersh S, Tolmachev AA, Grygorenko OO. Synthesis of α-C-Stereochemically Pure Secondary Sulfonamides. J Org Chem 2022. [PMID: 35441519 DOI: 10.1021/acs.joc.2c00480] [Reference Citation Analysis]
48 Tereshchenko OD, Perebiynis MY, Knysh IV, Vasylets OV, Sorochenko AA, Slobodyanyuk EY, Rusanov EB, Borysov OV, Kolotilov SV, Ryabukhin SV, Volochnyuk DM. Electrochemical Scaled‐up Synthesis of Cyclic Enecarbamates as Starting Materials for Medicinal Chemistry Relevant Building Bocks. Adv Synth Catal 2020;362:3229-42. [DOI: 10.1002/adsc.202000450] [Cited by in Crossref: 5] [Cited by in F6Publishing: 3] [Article Influence: 2.5] [Reference Citation Analysis]