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Hassan AS, Morsy NM, Aboulthana WM, Ragab A. Exploring novel derivatives of isatin-based Schiff bases as multi-target agents: design, synthesis, in vitro biological evaluation, and in silico ADMET analysis with molecular modeling simulations. RSC Adv 2023;13:9281-303. [PMID: 36950709 DOI: 10.1039/d3ra00297g] [Reference Citation Analysis]
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Ayman R, Abusaif MS, Radwan AM, Elmetwally AM, Ragab A. Development of novel pyrazole, imidazo[1,2-b]pyrazole, and pyrazolo[1,5-a]pyrimidine derivatives as a new class of COX-2 inhibitors with immunomodulatory potential. Eur J Med Chem 2023;249:115138. [PMID: 36696764 DOI: 10.1016/j.ejmech.2023.115138] [Reference Citation Analysis]
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Ragab A, Abusaif MS, Gohar NA, Aboul-Magd DS, Fayed EA, Ammar YA. Development of new spiro[1,3]dithiine-4,11'-indeno[1,2-b]quinoxaline derivatives as S. aureus Sortase A inhibitors and radiosterilization with molecular modeling simulation. Bioorg Chem 2023;131:106307. [PMID: 36481380 DOI: 10.1016/j.bioorg.2022.106307] [Cited by in Crossref: 2] [Cited by in F6Publishing: 1] [Article Influence: 2.0] [Reference Citation Analysis]
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Hassan AS, Morsy NM, Aboulthana WM, Ragab A. In vitro enzymatic evaluation of some pyrazolo[1,5-a]pyrimidine derivatives: Design, synthesis, antioxidant, anti-diabetic, anti-Alzheimer, and anti-arthritic activities with molecular modeling simulation. Drug Dev Res 2023;84:3-24. [PMID: 36380556 DOI: 10.1002/ddr.22008] [Cited by in Crossref: 1] [Cited by in F6Publishing: 1] [Article Influence: 1.0] [Reference Citation Analysis]
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Gul M, Turk Celikoglu E, Idil O, Tas G, Pelit E. Synthesis, antimicrobial activity and molecular docking studies of spiroquinoline-indoline-dione and spiropyrazolo-indoline-dione derivatives. Sci Rep 2023;13:1676. [PMID: 36717728 DOI: 10.1038/s41598-023-27777-z] [Reference Citation Analysis]
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Ragab A, Fouad SA, Ammar YA, Aboul-Magd DS, Abusaif MS. Antibiofilm and Anti-Quorum-Sensing Activities of Novel Pyrazole and Pyrazolo[1,5-a]pyrimidine Derivatives as Carbonic Anhydrase I and II Inhibitors: Design, Synthesis, Radiosterilization, and Molecular Docking Studies. Antibiotics (Basel) 2023;12. [PMID: 36671329 DOI: 10.3390/antibiotics12010128] [Cited by in Crossref: 1] [Article Influence: 1.0] [Reference Citation Analysis]
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