1 |
Ling X, Liu S, Yang Y, Dong Q, Marcaurelle LA, Huang W, Ding Y, Wang X, Lu X. Modular Click Assembly DNA-Encoded Glycoconjugate Libraries with on-DNA Functional Group Transformations. Bioconjug Chem 2023. [PMID: 36961996 DOI: 10.1021/acs.bioconjchem.3c00068] [Reference Citation Analysis]
|
2 |
Fang X, Liao H, Fan X, Wang Y, Wang H, Zhang G, Fang W, Li Y, Li Y. Incorporation of viridicatin alkaloid-like scaffolds into DNA-encoded chemical libraries. Org Biomol Chem 2023;21:2162-6. [PMID: 36799438 DOI: 10.1039/d2ob02278h] [Reference Citation Analysis]
|
3 |
Zhao G, Wang H, Luo J, He X, Xiong F, Li Y, Zhang G, Li Y. Multicomponent DNA-Compatible Synthesis of an Annelated Benzodiazepine Scaffold for Focused Chemical Libraries. Org Lett 2023;25:665-70. [PMID: 36693020 DOI: 10.1021/acs.orglett.2c04293] [Reference Citation Analysis]
|
4 |
Montoya AL, Glavatskikh M, Halverson BJ, Yuen LH, Schüler H, Kireev D, Franzini RM. Combining pharmacophore models derived from DNA-encoded chemical libraries with structure-based exploration to predict Tankyrase 1 inhibitors. Eur J Med Chem 2023;246:114980. [PMID: 36495630 DOI: 10.1016/j.ejmech.2022.114980] [Reference Citation Analysis]
|
5 |
Nie Q, Sun J, Fang X, He X, Xiong F, Zhang G, Li Y, Li Y. Antimony salt-promoted cyclization facilitating on-DNA syntheses of dihydroquinazolinone derivatives and its applications. Chinese Chemical Letters 2023. [DOI: 10.1016/j.cclet.2023.108132] [Reference Citation Analysis]
|
6 |
Xiong F, Xu H, Yu M, Chen X, Zhong Z, Guo Y, Chen M, Ou H, Wu J, Xie A, Xiong J, Xu L, Zhang L, Zhong Q, Huang L, Li Z, Zhang T, Jin F, He X. 3CLpro inhibitors: DEL-based molecular generation. Front Pharmacol 2022;13:1085665. [PMID: 36569316 DOI: 10.3389/fphar.2022.1085665] [Reference Citation Analysis]
|
7 |
Gao Y, Sun Y, Zhao G, Zhang G, Li Y, Li Y. On-DNA Synthesis of Functionalized 4H-Pyran Scaffolds for Focused DNA-Encoded Chemical Libraries. Org Lett 2022. [PMID: 36053053 DOI: 10.1021/acs.orglett.2c02714] [Reference Citation Analysis]
|
8 |
Xu H, Tan T, Zhang Y, Wang Y, Pan K, Yao Y, Zhang S, Gu Y, Chen W, Li J, Dong H, Meng Y, Ma P, Hou W, Yang G. Metal‐Free and Open‐Air Arylation Reactions of Diaryliodonium Salts for DNA‐Encoded Library Synthesis. Advanced Science. [DOI: 10.1002/advs.202202790] [Cited by in F6Publishing: 1] [Reference Citation Analysis]
|
9 |
Sun J, Nie Q, Fang X, He Z, Zhang G, Li Y, Li Y. Vinyl azide as a synthon for DNA-compatible divergent transformations into N-heterocycles. Org Biomol Chem 2022;20:5045-9. [PMID: 35703385 DOI: 10.1039/d2ob00862a] [Cited by in Crossref: 1] [Cited by in F6Publishing: 2] [Article Influence: 1.0] [Reference Citation Analysis]
|
10 |
Siripuram VK, Sunkari YK, Nguyen T, Flajolet M. DNA-Compatible Suzuki-Miyaura Cross-Coupling Reaction of Aryl Iodides With (Hetero)Aryl Boronic Acids for DNA-Encoded Libraries. Front Chem 2022;10:894603. [DOI: 10.3389/fchem.2022.894603] [Cited by in Crossref: 1] [Cited by in F6Publishing: 1] [Article Influence: 1.0] [Reference Citation Analysis]
|
11 |
Fang X, Wang Y, He P, Liao H, Zhang G, Li Y, Li Y. Visible Light-Promoted Divergent Benzoheterocyclization from Aldehydes for DNA-Encoded Chemical Libraries. Org Lett 2022. [PMID: 35467894 DOI: 10.1021/acs.orglett.2c01187] [Cited by in Crossref: 4] [Cited by in F6Publishing: 5] [Article Influence: 4.0] [Reference Citation Analysis]
|
12 |
Yang J, Xia S, Liu J, Yu Z, Mei L, Lu W, Chen Y, Chen S, Wang X, Lu X. DNA-Encoded Focused Indazole Library Synthesis by a Palladium-Mediated C-N(sp2) Cross-Coupling Reaction between DNA-linked (hetero)aryl halides and Aromatic Nitrogen Heterocycles. Tetrahedron Letters 2022. [DOI: 10.1016/j.tetlet.2022.153732] [Reference Citation Analysis]
|
13 |
Li X, Zhang J, Liu C, Sun J, Li Y, Zhang G, Li Y. Aryl diazonium intermediates enable mild DNA-compatible C–C bond formation for medicinally relevant combinatorial library synthesis. Chem Sci 2022. [DOI: 10.1039/d2sc04482j] [Reference Citation Analysis]
|
14 |
Gao Y, Sun Y, Fang X, Zhao G, Li X, Zhang G, Li Y, Li Y. Development of on-DNA vinyl sulfone synthesis for DNA-encoded chemical libraries. Org Chem Front . [DOI: 10.1039/d2qo00881e] [Cited by in Crossref: 1] [Cited by in F6Publishing: 3] [Article Influence: 1.0] [Reference Citation Analysis]
|