| 1 |
Li L, Matsuo B, Levitre G, McClain EJ, Voight EA, Crane EA, Molander GA. Dearomative intermolecular [2 + 2] photocycloaddition for construction of C(sp(3))-rich heterospirocycles on-DNA. Chem Sci 2023;14:2713-20. [PMID: 36908969 DOI: 10.1039/d3sc00144j] [Reference Citation Analysis]
|
| 2 |
Mantell MA, Marcaurelle L, Ding Y. One Reaction Served Three Ways: The On-DNA Ugi 4C-3C Reaction for the Formation of Lactams. Org Lett 2023;25:1241-5. [PMID: 36802674 DOI: 10.1021/acs.orglett.2c04043] [Reference Citation Analysis]
|
| 3 |
Krishna Sunkari Y, Kumar Siripuram V, Flajolet M. Diversity-Oriented Synthesis (DOS) of On-DNA Peptidomimetics from Acid-Derived Phosphonium Ylides. Chemistry 2023;29:e202203037. [PMID: 36653313 DOI: 10.1002/chem.202203037] [Reference Citation Analysis]
|
| 4 |
Matsuo B, Granados A, Levitre G, Molander GA. Photochemical Methods Applied to DNA Encoded Library (DEL) Synthesis. Acc Chem Res 2023;56:385-401. [PMID: 36656960 DOI: 10.1021/acs.accounts.2c00778] [Reference Citation Analysis]
|
| 5 |
Chheda PR, Simmons N, Schuman DP, Shi Z. Photoredox-Mediated Deoxygenative Alkylation of DNA-Tagged Alkenes with Activated Alcohols. Org Lett 2022;24:9514-9. [PMID: 36541781 DOI: 10.1021/acs.orglett.2c03994] [Reference Citation Analysis]
|
| 6 |
Osawa T, Ren Q, Obika S. Development of Phosphoramidite Reagents for the Synthesis of Base-Labile Oligonucleotides Modified with a Linear Aminoalkyl and Amino-PEG Linker at the 3'-End. Molecules 2022;27. [PMID: 36500594 DOI: 10.3390/molecules27238501] [Reference Citation Analysis]
|
| 7 |
Young RJ, Flitsch SL, Grigalunas M, Leeson PD, Quinn RJ, Turner NJ, Waldmann H. The Time and Place for Nature in Drug Discovery. JACS Au 2022;2:2400-2416. [DOI: 10.1021/jacsau.2c00415] [Reference Citation Analysis]
|
| 8 |
Zwillinger M, Fischer L, Sályi G, Szabó S, Csékei M, Huc I, Kotschy A. Isotope Ratio Encoding of Sequence-Defined Oligomers. J Am Chem Soc 2022. [PMID: 36206533 DOI: 10.1021/jacs.2c08135] [Reference Citation Analysis]
|
| 9 |
Sun Z, Zhang J, Zhang H, Cao H, Xiao L, Yang K, Hu YJ. DNA Compatible Oxidization and Amidation of Terminal Alkynes. Bioconjug Chem 2022. [PMID: 36001094 DOI: 10.1021/acs.bioconjchem.2c00340] [Reference Citation Analysis]
|
| 10 |
Luo A, Zhang Z, Zeng F, Wang X, Zhao X, Yang K, Hu YJ. Kinugasa Reaction for DNA-Encoded β-Lactam Library Synthesis. Org Lett 2022. [PMID: 35916753 DOI: 10.1021/acs.orglett.2c02237] [Cited by in Crossref: 1] [Cited by in F6Publishing: 1] [Article Influence: 1.0] [Reference Citation Analysis]
|
| 11 |
Sun J, Nie Q, Fang X, He Z, Zhang G, Li Y, Li Y. Vinyl azide as a synthon for DNA-compatible divergent transformations into N-heterocycles. Org Biomol Chem 2022;20:5045-9. [PMID: 35703385 DOI: 10.1039/d2ob00862a] [Cited by in Crossref: 1] [Cited by in F6Publishing: 2] [Article Influence: 1.0] [Reference Citation Analysis]
|
| 12 |
Siripuram VK, Sunkari YK, Nguyen T, Flajolet M. DNA-Compatible Suzuki-Miyaura Cross-Coupling Reaction of Aryl Iodides With (Hetero)Aryl Boronic Acids for DNA-Encoded Libraries. Front Chem 2022;10:894603. [DOI: 10.3389/fchem.2022.894603] [Cited by in Crossref: 1] [Cited by in F6Publishing: 1] [Article Influence: 1.0] [Reference Citation Analysis]
|
| 13 |
Bajusz D, Keserű GM. Maximizing the integration of virtual and experimental screening in hit discovery. Expert Opin Drug Discov 2022;:1-12. [PMID: 35671403 DOI: 10.1080/17460441.2022.2085685] [Reference Citation Analysis]
|
| 14 |
Fang X, Wang Y, He P, Liao H, Zhang G, Li Y, Li Y. Visible Light-Promoted Divergent Benzoheterocyclization from Aldehydes for DNA-Encoded Chemical Libraries. Org Lett 2022. [PMID: 35467894 DOI: 10.1021/acs.orglett.2c01187] [Cited by in Crossref: 4] [Cited by in F6Publishing: 5] [Article Influence: 4.0] [Reference Citation Analysis]
|
| 15 |
Cai K, Ran Y, Sun W, Gao S, Li J, Wan J, Liu G. Palladium-Mediated Hydroamination of DNA-Conjugated Aryl Alkenes. Front Chem 2022;10:851674. [DOI: 10.3389/fchem.2022.851674] [Reference Citation Analysis]
|
| 16 |
Shen Y, Yang G, Huang W, Shaginian A, Lin Q, Wan J, Li J, Deng Y, Liu G. Photoredox Deaminative Alkylation in DNA-Encoded Library Synthesis. Org Lett 2022. [PMID: 35362987 DOI: 10.1021/acs.orglett.2c00697] [Cited by in Crossref: 5] [Cited by in F6Publishing: 6] [Article Influence: 5.0] [Reference Citation Analysis]
|
| 17 |
Pei H, Guo W, Peng Y, Xiong H, Chen Y. Targeting key proteins involved in transcriptional regulation for cancer therapy: Current strategies and future prospective. Med Res Rev 2022. [PMID: 35312190 DOI: 10.1002/med.21886] [Cited by in Crossref: 4] [Cited by in F6Publishing: 6] [Article Influence: 4.0] [Reference Citation Analysis]
|
| 18 |
Zhao G, Zhong S, Zhang G, Li Y, Li Y. Reversible Covalent Headpiece Enables Interconversion between Double‐ and Single‐Stranded DNA‐Encoded Chemical Libraries. Angewandte Chemie 2022;134. [DOI: 10.1002/ange.202115157] [Cited by in Crossref: 1] [Cited by in F6Publishing: 1] [Article Influence: 1.0] [Reference Citation Analysis]
|
| 19 |
Nie Q, Fang X, Liu C, Zhang G, Fan X, Li Y, Li Y. DNA-Compatible ortho -Phthalaldehyde (OPA)-Mediated 2-Substituted Isoindole Core Formation and Applications. J Org Chem . [DOI: 10.1021/acs.joc.1c02496] [Cited by in Crossref: 6] [Cited by in F6Publishing: 7] [Article Influence: 6.0] [Reference Citation Analysis]
|
| 20 |
Zhong S, Fang X, Wang Y, Zhang G, Li Y, Li Y. DNA-Compatible Diversification of Indole π-Activated Alcohols via a Direct Dehydrative Coupling Strategy. Org Lett 2022. [PMID: 35050627 DOI: 10.1021/acs.orglett.1c04169] [Cited by in Crossref: 6] [Cited by in F6Publishing: 7] [Article Influence: 6.0] [Reference Citation Analysis]
|
| 21 |
Kita R, Osawa T, Obika S. Conjugation of oligonucleotides with activated carbamate reagents prepared by the Ugi reaction for oligonucleotide library synthesis. RSC Chem Biol . [DOI: 10.1039/d1cb00240f] [Reference Citation Analysis]
|
| 22 |
Anderson MJ, Castan IFSF, Graham JS, Hassan H, Odger J, Salvini CLA, Taylor C, Waring MJ. Advancements in DEL-Compatible Chemical Reactions. Topics in Medicinal Chemistry 2022. [DOI: 10.1007/7355_2022_151] [Reference Citation Analysis]
|
| 23 |
Zhu H, Montgomery JI, Stanton RV. Cheminformatics Approaches Aiding the Design and Selection of DNA-Encoded Libraries. Topics in Medicinal Chemistry 2022. [DOI: 10.1007/7355_2022_148] [Reference Citation Analysis]
|
| 24 |
Krumb M, Kammer LM, Badir SO, Cabrera-afonso MJ, Wu VE, Huang M, Csakai A, Marcaurelle LA, Molander GA. Photochemical C–H arylation of heteroarenes for DNA-encoded library synthesis. Chem Sci . [DOI: 10.1039/d1sc05683b] [Cited by in Crossref: 13] [Cited by in F6Publishing: 13] [Article Influence: 13.0] [Reference Citation Analysis]
|
| 25 |
Gui Y, Li X. Selection Strategies in DNA-Encoded Libraries. Topics in Medicinal Chemistry 2022. [DOI: 10.1007/7355_2022_149] [Reference Citation Analysis]
|
| 26 |
Marcaurelle L, Tear W, Yao G. From DEL Selections to Validated Hits to Clinical Leads. Topics in Medicinal Chemistry 2022. [DOI: 10.1007/7355_2022_150] [Reference Citation Analysis]
|
| 27 |
Li X, Zhang J, Liu C, Sun J, Li Y, Zhang G, Li Y. Aryl diazonium intermediates enable mild DNA-compatible C–C bond formation for medicinally relevant combinatorial library synthesis. Chem Sci 2022. [DOI: 10.1039/d2sc04482j] [Reference Citation Analysis]
|
| 28 |
Gao Y, Sun Y, Fang X, Zhao G, Li X, Zhang G, Li Y, Li Y. Development of on-DNA vinyl sulfone synthesis for DNA-encoded chemical libraries. Org Chem Front . [DOI: 10.1039/d2qo00881e] [Cited by in Crossref: 1] [Cited by in F6Publishing: 3] [Article Influence: 1.0] [Reference Citation Analysis]
|
| 29 |
Gao Y, Zhao G, He P, Zhang G, Li Y, Li Y. DNA-Compatible Synthesis of α,β-Epoxyketones for DNA-Encoded Chemical Libraries. Bioconjug Chem 2021. [PMID: 34927428 DOI: 10.1021/acs.bioconjchem.1c00567] [Cited by in Crossref: 7] [Cited by in F6Publishing: 7] [Article Influence: 3.5] [Reference Citation Analysis]
|
| 30 |
Zhao G, Zhong S, Zhang G, Li Y, Li Y. Reversible Covalent Headpiece Enables Interconversion between Double- and Single-Stranded DNA-Encoded Chemical Libraries. Angew Chem Int Ed Engl 2021;:e202115157. [PMID: 34904335 DOI: 10.1002/anie.202115157] [Cited by in Crossref: 8] [Cited by in F6Publishing: 10] [Article Influence: 4.0] [Reference Citation Analysis]
|
| 31 |
Fair RJ, Walsh RT, Hupp CD. The expanding reaction toolkit for DNA-encoded libraries. Bioorg Med Chem Lett 2021;51:128339. [PMID: 34478840 DOI: 10.1016/j.bmcl.2021.128339] [Cited by in Crossref: 16] [Cited by in F6Publishing: 18] [Article Influence: 8.0] [Reference Citation Analysis]
|
| 32 |
Nie Q, Zhong S, Li Y, Zhang G, Li Y. Second-generation DNA-encoded multiple display on a constant macrocyclic scaffold enabled by an orthogonal protecting group strategy. Chinese Chemical Letters 2021. [DOI: 10.1016/j.cclet.2021.09.041] [Cited by in Crossref: 8] [Cited by in F6Publishing: 8] [Article Influence: 4.0] [Reference Citation Analysis]
|
| 33 |
Silvestri IP, Colbon PJJ. The Growing Importance of Chirality in 3D Chemical Space Exploration and Modern Drug Discovery Approaches for Hit-ID: Topical Innovations. ACS Med Chem Lett 2021;12:1220-9. [PMID: 34413951 DOI: 10.1021/acsmedchemlett.1c00251] [Cited by in Crossref: 6] [Cited by in F6Publishing: 7] [Article Influence: 3.0] [Reference Citation Analysis]
|
