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Quancard J, Vulpetti A, Bach A, Cox B, Guéret SM, Hartung IV, Koolman HF, Laufer S, Messinger J, Sbardella G, Craft R. The European Federation for Medicinal Chemistry and Chemical Biology (EFMC) Best Practice Initiative: Hit Generation. ChemMedChem 2023;:e202300002. [PMID: 36892096 DOI: 10.1002/cmdc.202300002] [Reference Citation Analysis]
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Fang X, Liao H, Fan X, Wang Y, Wang H, Zhang G, Fang W, Li Y, Li Y. Incorporation of viridicatin alkaloid-like scaffolds into DNA-encoded chemical libraries. Org Biomol Chem 2023;21:2162-6. [PMID: 36799438 DOI: 10.1039/d2ob02278h] [Reference Citation Analysis]
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Li L, Matsuo B, Levitre G, McClain EJ, Voight EA, Crane EA, Molander GA. Dearomative intermolecular [2 + 2] photocycloaddition for construction of C(sp(3))-rich heterospirocycles on-DNA. Chem Sci 2023;14:2713-20. [PMID: 36908969 DOI: 10.1039/d3sc00144j] [Reference Citation Analysis]
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Mantell MA, Marcaurelle L, Ding Y. One Reaction Served Three Ways: The On-DNA Ugi 4C-3C Reaction for the Formation of Lactams. Org Lett 2023;25:1241-5. [PMID: 36802674 DOI: 10.1021/acs.orglett.2c04043] [Reference Citation Analysis]
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Dockerill M, Winssinger N. DNA-Encoded Libraries: Towards Harnessing their Full Power with Darwinian Evolution. Angew Chem Int Ed Engl 2023;62:e202215542. [PMID: 36458812 DOI: 10.1002/anie.202215542] [Cited by in Crossref: 2] [Cited by in F6Publishing: 2] [Article Influence: 2.0] [Reference Citation Analysis]
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Modukuri RK, Monsivais D, Li F, Palaniappan M, Bohren KM, Tan Z, Ku AF, Wang Y, Madasu C, Li JY, Tang S, Miklossy G, Palmer SS, Young DW, Matzuk MM. Discovery of Highly Potent and BMPR2-Selective Kinase Inhibitors Using DNA-Encoded Chemical Library Screening. J Med Chem 2023;66:2143-60. [PMID: 36719862 DOI: 10.1021/acs.jmedchem.2c01886] [Reference Citation Analysis]
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Cai B, Mhetre AB, Krusemark CJ. Selection methods for proximity-dependent enrichment of ligands from DNA-encoded libraries using enzymatic fusion proteins. Chem Sci 2023;14:245-50. [PMID: 36687357 DOI: 10.1039/d2sc05495g] [Reference Citation Analysis]
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Luo A, Zhou H, Zhou Q, Hua Q, Zhao X, Yu X, Yang K, Hu YJ. On-DNA Alkyne Iodination and Acetylenic Coupling as a Useful Tool for DEL Synthesis. Bioconjug Chem 2022;33:2299-306. [PMID: 36450158 DOI: 10.1021/acs.bioconjchem.2c00471] [Reference Citation Analysis]
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Press WH. Fast trimer statistics facilitate accurate decoding of large random DNA barcode sets even at large sequencing error rates. PNAS Nexus 2022;1:pgac252. [PMID: 36712375 DOI: 10.1093/pnasnexus/pgac252] [Reference Citation Analysis]
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Blay V, Li X, Gerlach J, Urbina F, Ekins S. Combining DELs and machine learning for toxicology prediction. Drug Discov Today 2022;27:103351. [PMID: 36096360 DOI: 10.1016/j.drudis.2022.103351] [Cited by in Crossref: 1] [Article Influence: 1.0] [Reference Citation Analysis]
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Chen M, Zhu Z, Wisniewski T, Zhang X, Mclaren DG, Weinglass A, Saldanha SA. Label-free LC-MS based assay to characterize small molecule compound binding to cells. SLAS Discovery 2022. [DOI: 10.1016/j.slasd.2022.08.005] [Reference Citation Analysis]
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Sun Z, Zhang J, Zhang H, Cao H, Xiao L, Yang K, Hu YJ. DNA Compatible Oxidization and Amidation of Terminal Alkynes. Bioconjug Chem 2022. [PMID: 36001094 DOI: 10.1021/acs.bioconjchem.2c00340] [Reference Citation Analysis]
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Götte K, Dinter R, Justen L, Kockmann N, Brunschweiger A. Development of an Automatable Affinity Purification Process for DNA-Encoded Chemistry. ACS Omega. [DOI: 10.1021/acsomega.2c02906] [Reference Citation Analysis]
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Potowski M, Kunig VBK, Eberlein L, Škopić MK, Vakalopoulos A, Kast SM, Brunschweiger A. Investigations Into Chemically Stabilized Four-Letter DNA for DNA-Encoded Chemistry. Front Chem 2022;10:894563. [PMID: 35755251 DOI: 10.3389/fchem.2022.894563] [Reference Citation Analysis]
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Gui Y, Wong CS, Zhao G, Xie C, Hou R, Li Y, Li G, Li X. Converting Double-Stranded DNA-Encoded Libraries (DELs) to Single-Stranded Libraries for More Versatile Selections. ACS Omega 2022;7:11491-500. [PMID: 35415338 DOI: 10.1021/acsomega.2c01152] [Cited by in Crossref: 3] [Cited by in F6Publishing: 3] [Article Influence: 3.0] [Reference Citation Analysis]
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Shen Y, Yang G, Huang W, Shaginian A, Lin Q, Wan J, Li J, Deng Y, Liu G. Photoredox Deaminative Alkylation in DNA-Encoded Library Synthesis. Org Lett 2022. [PMID: 35362987 DOI: 10.1021/acs.orglett.2c00697] [Cited by in Crossref: 5] [Cited by in F6Publishing: 6] [Article Influence: 5.0] [Reference Citation Analysis]
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Yang J, Xia S, Liu J, Yu Z, Mei L, Lu W, Chen Y, Chen S, Wang X, Lu X. DNA-Encoded Focused Indazole Library Synthesis by a Palladium-Mediated C-N(sp2) Cross-Coupling Reaction between DNA-linked (hetero)aryl halides and Aromatic Nitrogen Heterocycles. Tetrahedron Letters 2022. [DOI: 10.1016/j.tetlet.2022.153732] [Reference Citation Analysis]
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Chines S, Ehrt C, Potowski M, Biesenkamp F, Grützbach L, Brunner S, van den Broek F, Bali S, Ickstadt K, Brunschweiger A. Navigating chemical reaction space – application to DNA-encoded chemistry. Chem Sci 2022;13:11221-31. [DOI: 10.1039/d2sc02474h] [Reference Citation Analysis]
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