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For: Baxter CA, Cleator E, Brands KMJ, Edwards JS, Reamer RA, Sheen FJ, Stewart GW, Strotman NA, Wallace DJ. The First Large-Scale Synthesis of MK-4305: A Dual Orexin Receptor Antagonist for the Treatment of Sleep Disorder. Org Process Res Dev 2011;15:367-75. [DOI: 10.1021/op1002853] [Cited by in Crossref: 70] [Cited by in F6Publishing: 44] [Article Influence: 6.4] [Reference Citation Analysis]
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17 Strotman NA, Baxter CA, Brands KM, Cleator E, Krska SW, Reamer RA, Wallace DJ, Wright TJ. Reaction development and mechanistic study of a ruthenium catalyzed intramolecular asymmetric reductive amination en route to the dual Orexin inhibitor Suvorexant (MK-4305). J Am Chem Soc 2011;133:8362-71. [PMID: 21528938 DOI: 10.1021/ja202358f] [Cited by in Crossref: 86] [Cited by in F6Publishing: 61] [Article Influence: 7.8] [Reference Citation Analysis]
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26 Teci M, Tilley M, Mcguire MA, Organ MG. Handling Hazards Using Continuous Flow Chemistry: Synthesis of N1 -Aryl-[1,2,3]-triazoles from Anilines via Telescoped Three-Step Diazotization, Azidodediazotization, and [3 + 2] Dipolar Cycloaddition Processes. Org Process Res Dev 2016;20:1967-73. [DOI: 10.1021/acs.oprd.6b00292] [Cited by in Crossref: 40] [Cited by in F6Publishing: 19] [Article Influence: 6.7] [Reference Citation Analysis]
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30 Gupta S, Chandna N, Singh AK, Jain N. Regioselective Synthesis of N2-Alkylated-1,2,3 Triazoles and N1-Alkylated Benzotriazoles: Cu2S as a Recyclable Nanocatalyst for Oxidative Amination of N, N-Dimethylbenzylamines. J Org Chem 2018;83:3226-35. [PMID: 29463081 DOI: 10.1021/acs.joc.8b00107] [Cited by in Crossref: 13] [Cited by in F6Publishing: 7] [Article Influence: 3.3] [Reference Citation Analysis]
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