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For: Gironda-Martínez A, Donckele EJ, Samain F, Neri D. DNA-Encoded Chemical Libraries: A Comprehensive Review with Succesful Stories and Future Challenges. ACS Pharmacol Transl Sci 2021;4:1265-79. [PMID: 34423264 DOI: 10.1021/acsptsci.1c00118] [Cited by in Crossref: 30] [Cited by in F6Publishing: 35] [Article Influence: 15.0] [Reference Citation Analysis]
Number Citing Articles
1 Sun Z, Xiao L, Chen Y, Wang J, Zeng F, Zhang H, Zhang J, Yang K, Hu YJ. Constructive On-DNA Abramov Reaction and Pudovik Reaction for DEL Synthesis. ACS Med Chem Lett 2023. [DOI: 10.1021/acsmedchemlett.3c00022] [Reference Citation Analysis]
2 Luo A, Zhou H, Hua Q, An Y, Ma H, Zhao X, Yang K, Hu YJ. Development of the Inverse Sonogashira Reaction for DEL Synthesis. ACS Med Chem Lett 2023;14:270-7. [PMID: 36923912 DOI: 10.1021/acsmedchemlett.2c00477] [Cited by in Crossref: 1] [Article Influence: 1.0] [Reference Citation Analysis]
3 Quancard J, Vulpetti A, Bach A, Cox B, Guéret SM, Hartung IV, Koolman HF, Laufer S, Messinger J, Sbardella G, Craft R. The European Federation for Medicinal Chemistry and Chemical Biology (EFMC) Best Practice Initiative: Hit Generation. ChemMedChem 2023;:e202300002. [PMID: 36892096 DOI: 10.1002/cmdc.202300002] [Reference Citation Analysis]
4 Stanway-Gordon HA, Odger JA, Waring MJ. Development of a Micellar-Promoted Heck Reaction for the Synthesis of DNA-Encoded Libraries. Bioconjug Chem 2023. [PMID: 36883323 DOI: 10.1021/acs.bioconjchem.3c00051] [Reference Citation Analysis]
5 Zhu KF, Yuan C, Du YM, Sun KL, Zhang XK, Vogel H, Jia XD, Gao YZ, Zhang QF, Wang DP, Zhang HW. Applications and prospects of cryo-EM in drug discovery. Mil Med Res 2023;10:10. [PMID: 36872349 DOI: 10.1186/s40779-023-00446-y] [Reference Citation Analysis]
6 Mantell MA, Marcaurelle L, Ding Y. One Reaction Served Three Ways: The On-DNA Ugi 4C-3C Reaction for the Formation of Lactams. Org Lett 2023;25:1241-5. [PMID: 36802674 DOI: 10.1021/acs.orglett.2c04043] [Reference Citation Analysis]
7 Sala D, Batebi H, Ledwitch K, Hildebrand PW, Meiler J. Targeting in silico GPCR conformations with ultra-large library screening for hit discovery. Trends Pharmacol Sci 2023;44:150-61. [PMID: 36669974 DOI: 10.1016/j.tips.2022.12.006] [Cited by in Crossref: 1] [Cited by in F6Publishing: 1] [Article Influence: 1.0] [Reference Citation Analysis]
8 Mahdavi-Amiri Y, Hu MSJ, Frias N, Movahedi M, Csakai A, Marcaurelle LA, Hili R. Photoredox-catalysed hydroaminoalkylation of on-DNA N-arylamines. Org Biomol Chem 2023;21:1463-7. [PMID: 36655521 DOI: 10.1039/d2ob01956f] [Reference Citation Analysis]
9 Chan WC, Liu X, Magin RS, Girardi NM, Ficarro SB, Hu W, Tarazona Guzman MI, Starnbach CA, Felix A, Adelmant G, Varca AC, Hu B, Bratt AS, DaSilva E, Schauer NJ, Jaen Maisonet I, Dolen EK, Ayala AX, Marto JA, Buhrlage SJ. Accelerating inhibitor discovery for deubiquitinating enzymes. Nat Commun 2023;14:686. [PMID: 36754960 DOI: 10.1038/s41467-023-36246-0] [Reference Citation Analysis]
10 Chakravarty A, Yang PL. Targeted protein degradation as an antiviral approach. Antiviral Res 2023;210:105480. [PMID: 36567024 DOI: 10.1016/j.antiviral.2022.105480] [Reference Citation Analysis]
11 Duran-Frigola M, Cigler M, Winter GE. Advancing Targeted Protein Degradation via Multiomics Profiling and Artificial Intelligence. J Am Chem Soc 2023;145:2711-32. [PMID: 36706315 DOI: 10.1021/jacs.2c11098] [Reference Citation Analysis]
12 Cai B, Mhetre AB, Krusemark CJ. Selection methods for proximity-dependent enrichment of ligands from DNA-encoded libraries using enzymatic fusion proteins. Chem Sci 2023;14:245-50. [PMID: 36687357 DOI: 10.1039/d2sc05495g] [Reference Citation Analysis]
13 Miller S, Moos W, Munk B, Munk S, Hart C, Spellmeyer D. Drug discovery: Standing on the shoulders of giants. Managing the Drug Discovery Process 2023. [DOI: 10.1016/b978-0-12-824304-6.00001-8] [Reference Citation Analysis]
14 Miller S, Moos W, Munk B, Munk S, Hart C, Spellmeyer D. Drug discovery processes: When and where the rubber meets the road. Managing the Drug Discovery Process 2023. [DOI: 10.1016/b978-0-12-824304-6.00025-0] [Reference Citation Analysis]
15 Tunjic TM, Weber N, Brunsteiner M. Computer aided drug design in the development of proteolysis targeting chimeras. Computational and Structural Biotechnology Journal 2023;21:2058-2067. [DOI: 10.1016/j.csbj.2023.02.042] [Reference Citation Analysis]
16 Luo A, Zhou H, Zhou Q, Hua Q, Zhao X, Yu X, Yang K, Hu YJ. On-DNA Alkyne Iodination and Acetylenic Coupling as a Useful Tool for DEL Synthesis. Bioconjug Chem 2022;33:2299-306. [PMID: 36450158 DOI: 10.1021/acs.bioconjchem.2c00471] [Reference Citation Analysis]
17 Zhu H, Zhang Y, Li W, Huang N. A Comprehensive Survey of Prospective Structure-Based Virtual Screening for Early Drug Discovery in the Past Fifteen Years. Int J Mol Sci 2022;23. [PMID: 36555602 DOI: 10.3390/ijms232415961] [Reference Citation Analysis]
18 Osawa T, Ren Q, Obika S. Development of Phosphoramidite Reagents for the Synthesis of Base-Labile Oligonucleotides Modified with a Linear Aminoalkyl and Amino-PEG Linker at the 3'-End. Molecules 2022;27. [PMID: 36500594 DOI: 10.3390/molecules27238501] [Reference Citation Analysis]
19 Reverdy C, Gitton G, Guan X, Adhya I, Krishna Dumpati R, Roy S, Chall S, Ghosh A, Errasti G, Delacroix T, Chakrabarti R. Discovery of novel compounds as potent activators of Sirt3. Bioorganic & Medicinal Chemistry 2022;73:116999. [DOI: 10.1016/j.bmc.2022.116999] [Reference Citation Analysis]
20 Zhang Y, Xia S, Shi W, Lin B, Su X, Lu W, Wu X, Wang X, Lu X, Yan M, Zhang X. Radical C–H Sulfonation of Arenes: Its Applications on Bioactive and DNA-Encoded Molecules. Org Lett 2022. [DOI: 10.1021/acs.orglett.2c03077] [Reference Citation Analysis]
21 Furka Á. Forty years of combinatorial technology. Drug Discov Today 2022;27:103308. [PMID: 35760283 DOI: 10.1016/j.drudis.2022.06.008] [Cited by in Crossref: 1] [Cited by in F6Publishing: 1] [Article Influence: 1.0] [Reference Citation Analysis]
22 Janin YL. On drug discovery against infectious diseases and academic medicinal chemistry contributions. Beilstein J Org Chem 2022;18:1355-78. [DOI: 10.3762/bjoc.18.141] [Reference Citation Analysis]
23 Chana CK, Maisonneuve P, Posternak G, Grinberg NGA, Poirson J, Ona SM, Ceccarelli DF, Mader P, St-Cyr DJ, Pau V, Kurinov I, Tang X, Deng D, Cui W, Su W, Kuai L, Soll R, Tyers M, Röst HL, Batey RA, Taipale M, Gingras AC, Sicheri F. Discovery and Structural Characterization of Small Molecule Binders of the Human CTLH E3 Ligase Subunit GID4. J Med Chem 2022. [PMID: 36117290 DOI: 10.1021/acs.jmedchem.2c00509] [Reference Citation Analysis]
24 Sun Z, Zhang J, Zhang H, Cao H, Xiao L, Yang K, Hu YJ. DNA Compatible Oxidization and Amidation of Terminal Alkynes. Bioconjug Chem 2022. [PMID: 36001094 DOI: 10.1021/acs.bioconjchem.2c00340] [Reference Citation Analysis]
25 Sunkari YK, Meijer L, Flajolet M. The protein kinase CK1: Inhibition, activation, and possible allosteric modulation. Front Mol Biosci 2022;9:916232. [DOI: 10.3389/fmolb.2022.916232] [Reference Citation Analysis]
26 Yen-Pon E, Li L, Levitre G, Majhi J, McClain EJ, Voight EA, Crane EA, Molander GA. On-DNA Hydroalkylation to Introduce Diverse Bicyclo[1.1.1]pentanes and Abundant Alkyls via Halogen Atom Transfer. J Am Chem Soc 2022;144:12184-91. [PMID: 35759692 DOI: 10.1021/jacs.2c03025] [Cited by in Crossref: 5] [Cited by in F6Publishing: 4] [Article Influence: 5.0] [Reference Citation Analysis]
27 Eom S, Kwon T, Lee DY, Park CH, Kim HJ. Copper-Mediated Three-Component Reaction for the Synthesis of N-Acylsulfonamide on DNA. Org Lett 2022. [PMID: 35775977 DOI: 10.1021/acs.orglett.2c01675] [Reference Citation Analysis]
28 Proj M, Bozovičar K, Hrast M, Frlan R, Gobec S. DNA-encoded library screening on two validated enzymes of the peptidoglycan biosynthetic pathway. Bioorganic & Medicinal Chemistry Letters 2022. [DOI: 10.1016/j.bmcl.2022.128915] [Reference Citation Analysis]
29 Potowski M, Kunig VBK, Eberlein L, Škopić MK, Vakalopoulos A, Kast SM, Brunschweiger A. Investigations Into Chemically Stabilized Four-Letter DNA for DNA-Encoded Chemistry. Front Chem 2022;10:894563. [PMID: 35755251 DOI: 10.3389/fchem.2022.894563] [Reference Citation Analysis]
30 Bajusz D, Keserű GM. Maximizing the integration of virtual and experimental screening in hit discovery. Expert Opin Drug Discov 2022;:1-12. [PMID: 35671403 DOI: 10.1080/17460441.2022.2085685] [Reference Citation Analysis]
31 Ng TI, Correia I, Seagal J, Degoey DA, Schrimpf MR, Hardee DJ, Noey EL, Kati WM. Antiviral Drug Discovery for the Treatment of COVID-19 Infections. Viruses 2022;14:961. [DOI: 10.3390/v14050961] [Cited by in Crossref: 15] [Cited by in F6Publishing: 12] [Article Influence: 15.0] [Reference Citation Analysis]
32 Warr WA, Nicklaus MC, Nicolaou CA, Rarey M. Exploration of Ultralarge Compound Collections for Drug Discovery. J Chem Inf Model 2022. [PMID: 35421301 DOI: 10.1021/acs.jcim.2c00224] [Cited by in Crossref: 5] [Cited by in F6Publishing: 7] [Article Influence: 5.0] [Reference Citation Analysis]
33 Cai K, Ran Y, Sun W, Gao S, Li J, Wan J, Liu G. Palladium-Mediated Hydroamination of DNA-Conjugated Aryl Alkenes. Front Chem 2022;10:851674. [DOI: 10.3389/fchem.2022.851674] [Reference Citation Analysis]
34 Gui Y, Wong CS, Zhao G, Xie C, Hou R, Li Y, Li G, Li X. Converting Double-Stranded DNA-Encoded Libraries (DELs) to Single-Stranded Libraries for More Versatile Selections. ACS Omega 2022;7:11491-500. [PMID: 35415338 DOI: 10.1021/acsomega.2c01152] [Cited by in Crossref: 3] [Cited by in F6Publishing: 3] [Article Influence: 3.0] [Reference Citation Analysis]
35 Wu X, Zhang Q, Guo Y, Zhang H, Guo X, You Q, Wang L. Methods for the Discovery and Identification of Small Molecules Targeting Oxidative Stress-Related Protein–Protein Interactions: An Update. Antioxidants 2022;11:619. [DOI: 10.3390/antiox11040619] [Cited by in Crossref: 4] [Cited by in F6Publishing: 4] [Article Influence: 4.0] [Reference Citation Analysis]
36 Nicastri KA, Zappia S, Pratt JC, Duncan JM, Guzei IA, Fernández I, Schomaker JM. Tunable Aziridinium Ylide Reactivity: Non-covalent Interactions Enable Divergent Product Outcomes. ACS Catal 2022;12:1572-80. [PMID: 35291380 DOI: 10.1021/acscatal.1c05413] [Cited by in Crossref: 5] [Cited by in F6Publishing: 5] [Article Influence: 5.0] [Reference Citation Analysis]
37 Reverdy C, Gitton G, Guan X, Adhya I, Dumpati RK, Roy S, Chall S, Errasti G, Delacroix T, Chakrabarti R. Discovery of novel compounds as potent activators of Sirt3.. [DOI: 10.1101/2022.01.05.475007] [Reference Citation Analysis]
38 Ma H, Murray JB, Luo H, Cheng X, Chen Q, Song C, Duan C, Tan P, Zhang L, Liu J, Morgan BA, Li J, Wan J, Baker LM, Finnie W, Guetzoyan L, Harris R, Hendrickson N, Matassova N, Simmonite H, Smith J, Hubbard RE, Liu G. PAC-FragmentDEL – photoactivated covalent capture of DNA-encoded fragments for hit discovery. RSC Med Chem 2022. [DOI: 10.1039/d2md00197g] [Cited by in F6Publishing: 1] [Reference Citation Analysis]
39 Kita R, Osawa T, Obika S. Conjugation of oligonucleotides with activated carbamate reagents prepared by the Ugi reaction for oligonucleotide library synthesis. RSC Chem Biol . [DOI: 10.1039/d1cb00240f] [Reference Citation Analysis]
40 Zhu H, Montgomery JI, Stanton RV. Cheminformatics Approaches Aiding the Design and Selection of DNA-Encoded Libraries. Topics in Medicinal Chemistry 2022. [DOI: 10.1007/7355_2022_148] [Reference Citation Analysis]
41 Gui Y, Li X. Selection Strategies in DNA-Encoded Libraries. Topics in Medicinal Chemistry 2022. [DOI: 10.1007/7355_2022_149] [Reference Citation Analysis]
42 Morgan BA. A Perspective on 30 Years of DNA-Encoded Chemistry. Topics in Medicinal Chemistry 2022. [DOI: 10.1007/7355_2022_152] [Reference Citation Analysis]
43 Lessing A, Detta E, Scheuermann J, Brunschweiger A. Barcoding Strategies for the Synthesis of Genetically Encoded Chemical Libraries. Topics in Medicinal Chemistry 2022. [DOI: 10.1007/7355_2022_146] [Reference Citation Analysis]
44 Zhang Y, Franzini RM. Design Considerations in Constructing and Screening DNA-Encoded Libraries. Topics in Medicinal Chemistry 2022. [DOI: 10.1007/7355_2022_147] [Reference Citation Analysis]
45 Cochrane WG, Fitzgerald PR, Paegel BM. Antibacterial Discovery via Phenotypic DNA-Encoded Library Screening. ACS Chem Biol 2021;16:2752-6. [PMID: 34806373 DOI: 10.1021/acschembio.1c00714] [Cited by in Crossref: 1] [Cited by in F6Publishing: 3] [Article Influence: 0.5] [Reference Citation Analysis]
46 Gironda-Martínez A, Gorre ÉMD, Prati L, Gosalbes JF, Dakhel S, Cazzamalli S, Samain F, Donckele EJ, Neri D. Identification and Validation of New Interleukin-2 Ligands Using DNA-Encoded Libraries. J Med Chem 2021;64:17496-510. [PMID: 34821503 DOI: 10.1021/acs.jmedchem.1c01693] [Cited by in Crossref: 2] [Cited by in F6Publishing: 2] [Article Influence: 1.0] [Reference Citation Analysis]
47 Oehler S, Plais L, Bassi G, Neri D, Scheuermann J. Modular assembly and encoding strategies for dual-display DNA-encoded chemical libraries. Chem Commun (Camb) 2021;57:12289-92. [PMID: 34730584 DOI: 10.1039/d1cc04306d] [Cited by in Crossref: 3] [Cited by in F6Publishing: 4] [Article Influence: 1.5] [Reference Citation Analysis]
48 Furka Á. Combinatorial technology revitalized by DNA-encoding. MedComm (2020) 2021;2:481-9. [PMID: 34766157 DOI: 10.1002/mco2.84] [Cited by in Crossref: 2] [Cited by in F6Publishing: 4] [Article Influence: 1.0] [Reference Citation Analysis]
49 Fair RJ, Walsh RT, Hupp CD. The expanding reaction toolkit for DNA-encoded libraries. Bioorg Med Chem Lett 2021;51:128339. [PMID: 34478840 DOI: 10.1016/j.bmcl.2021.128339] [Cited by in Crossref: 16] [Cited by in F6Publishing: 18] [Article Influence: 8.0] [Reference Citation Analysis]