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Cited by in F6Publishing
For: Sakauchi N, Kohara Y, Sato A, Suzaki T, Imai Y, Okabe Y, Imai S, Saikawa R, Nagabukuro H, Kuno H, Fujita H, Kamo I, Yoshida M. Discovery of 5-Chloro-1-(5-chloro-2-(methylsulfonyl)benzyl)-2-imino-1,2-dihydropyridine-3-carboxamide (TAK-259) as a Novel, Selective, and Orally Active α 1D Adrenoceptor Antagonist with Antiurinary Frequency Effects: Reducing Human Ether-a-go-go-Related Gene (hERG) Liabilities. J Med Chem 2016;59:2989-3002. [DOI: 10.1021/acs.jmedchem.5b01528] [Cited by in Crossref: 5] [Cited by in F6Publishing: 5] [Article Influence: 0.8] [Reference Citation Analysis]
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1 Garrido A, Lepailleur A, Mignani SM, Dallemagne P, Rochais C. hERG toxicity assessment: Useful guidelines for drug design. Eur J Med Chem 2020;195:112290. [PMID: 32283295 DOI: 10.1016/j.ejmech.2020.112290] [Cited by in Crossref: 35] [Cited by in F6Publishing: 43] [Article Influence: 17.5] [Reference Citation Analysis]
2 Brown DG, Boström J. Where Do Recent Small Molecule Clinical Development Candidates Come From? J Med Chem 2018;61:9442-68. [DOI: 10.1021/acs.jmedchem.8b00675] [Cited by in Crossref: 86] [Cited by in F6Publishing: 90] [Article Influence: 21.5] [Reference Citation Analysis]
3 Ma D, Niu S, Zhao J, Jiang X, Jiang Y, Zhang X, Sun T. A New Class of Amide Ligands Enable Cu-Catalyzed Coupling of Sodium Methanesulfinate with (Hetero)aryl Chlorides: A New Class of Amide Ligands Enable Cu-Catalyzed Coupling of Sodium Methanesulfinate with (Hetero)aryl Chlorides. Chin J Chem 2017;35:1661-4. [DOI: 10.1002/cjoc.201700477] [Cited by in Crossref: 12] [Cited by in F6Publishing: 13] [Article Influence: 2.4] [Reference Citation Analysis]
4 Sakauchi N, Furukawa H, Shirai J, Sato A, Kuno H, Saikawa R, Yoshida M. Identification of 3,4-dihydro-2H-thiochromene 1,1-dioxide derivatives with a phenoxyethylamine group as highly potent and selective α1D adrenoceptor antagonists. Eur J Med Chem 2017;139:114-27. [PMID: 28800452 DOI: 10.1016/j.ejmech.2017.07.071] [Cited by in Crossref: 4] [Cited by in F6Publishing: 4] [Article Influence: 0.8] [Reference Citation Analysis]
5 Sato A, Sakauchi N, Shirai J, Furukawa H, Hara M, Miwa K, Fujita H, Miyamoto M, Tada N, Kuno H, Kameoka N, Maezaki H. Structure determination, synthesis, and biological evaluation of a metabolite of the selective α1D adrenoceptor antagonist TAK-259. Tetrahedron 2016;72:6334-6339. [DOI: 10.1016/j.tet.2016.08.013] [Reference Citation Analysis]