BPG is committed to discovery and dissemination of knowledge
Cited by in F6Publishing
For: Sun S, Fu J. Methyl-containing pharmaceuticals: Methylation in drug design. Bioorganic & Medicinal Chemistry Letters 2018;28:3283-9. [DOI: 10.1016/j.bmcl.2018.09.016] [Cited by in Crossref: 31] [Cited by in F6Publishing: 23] [Article Influence: 7.8] [Reference Citation Analysis]
Number Citing Articles
1 Liu D, Yu L, Yu Y, Xia Z, Song Z, Liao L, Tan Z, Chen X. Nickel-Catalyzed Ortho C-H Methylation of Aromatic Amides with Di- tert -butyl Peroxide as Methylation Reagent: Nickel-Catalyzed Ortho C-H Methylation of Aromatic Amides with Di- tert -butyl Peroxide as Methylation Reagent. Eur J Org Chem 2019;2019:6930-4. [DOI: 10.1002/ejoc.201901211] [Cited by in Crossref: 7] [Cited by in F6Publishing: 4] [Article Influence: 2.3] [Reference Citation Analysis]
2 Parcella K, Wang T, Eastman K, Zhang Z, Yin Z, Patel M, Tu Y, Zheng BZ, Walker MA, Saulnier MG, Frennesson D, Bowsher M, Gillis E, Peese K, Belema M, Cianci C, Dicker IB, Mcauliffe B, Ding B, Falk P, Simmermacher J, Parker DD, Sivaprakasam P, Kish K, Lewis H, Hanumegowda U, Jenkins S, Kadow JF, Krystal M, Meanwell NA, Naidu BN. Discovery and Preclinical Profiling of GSK3839919, a Potent HIV-1 Allosteric Integrase Inhibitor. ACS Med Chem Lett . [DOI: 10.1021/acsmedchemlett.2c00115] [Reference Citation Analysis]
3 Ding C, Ren Y, Sun C, Long J, Yin G. Regio- and Stereoselective Alkylboration of Endocyclic Olefins Enabled by Nickel Catalysis. J Am Chem Soc 2021;143:20027-34. [PMID: 34734714 DOI: 10.1021/jacs.1c09214] [Reference Citation Analysis]
4 Ramesh D, Sarkar D, Joji A, Singh M, Mohanty AK, G Vijayakumar B, Chatterjee M, Sriram D, Muthuvel SK, Kannan T. First-in-class pyrido[2,3-d]pyrimidine-2,4(1H,3H)-diones against leishmaniasis and tuberculosis: Rationale, in vitro, ex vivo studies and mechanistic insights. Arch Pharm (Weinheim) 2022;:e2100440. [PMID: 35106845 DOI: 10.1002/ardp.202100440] [Reference Citation Analysis]
5 Tsukamoto Y, Itoh S, Kobayashi M, Obora Y. Iridium-Catalyzed α-Methylation of α-Aryl Esters Using Methanol as the C1 Source. Org Lett 2019;21:3299-303. [DOI: 10.1021/acs.orglett.9b01025] [Cited by in Crossref: 14] [Cited by in F6Publishing: 7] [Article Influence: 4.7] [Reference Citation Analysis]
6 Templ J, Schnürch M. Selective α-Methylation of Aryl Ketones Using Quaternary Ammonium Salts as Solid Methylating Agents. J Org Chem . [DOI: 10.1021/acs.joc.1c03158] [Reference Citation Analysis]
7 Liu F, Ye ZP, Hu YZ, Gao J, Zheng L, Chen K, Xiang HY, Chen XQ, Yang H. N,N,N',N'-Tetramethylethylenediamine-Enabled Photoredox-Catalyzed C-H Methylation of N-Heteroarenes. J Org Chem 2021;86:11905-14. [PMID: 34344150 DOI: 10.1021/acs.joc.1c01325] [Reference Citation Analysis]
8 Guo YQ, Chen F, Deng CL, Zhang XG. Iodine-promoted ring-opening methylation of benzothiazoles with dimethyl sulfite. Chem Commun (Camb) 2021;57:1923-6. [PMID: 33496694 DOI: 10.1039/d0cc08096a] [Cited by in Crossref: 2] [Article Influence: 2.0] [Reference Citation Analysis]
9 Jin T, Xu L, Wang P, Hu X, Zhang R, Wu Z, Du W, Kan W, Li K, Wang C, Zhou Y, Li J, Liu T. Discovery and Development of a Potent, Selective, and Orally Bioavailable CHK1 Inhibitor Candidate: 5-((4-((3-Amino-3-methylbutyl)amino)-5-(trifluoromethyl)pyrimidin-2-yl)amino)picolinonitrile. J Med Chem 2021;64:15069-90. [PMID: 34665631 DOI: 10.1021/acs.jmedchem.1c00994] [Reference Citation Analysis]
10 Babbar P, Das P, Manickam Y, Mankad Y, Yadav S, Parvez S, Sharma A, Reddy DS. Design, Synthesis, and Structural Analysis of Cladosporin-Based Inhibitors of Malaria Parasites. ACS Infect Dis 2021;7:1777-94. [PMID: 33843204 DOI: 10.1021/acsinfecdis.1c00092] [Cited by in Crossref: 1] [Cited by in F6Publishing: 1] [Article Influence: 1.0] [Reference Citation Analysis]
11 Vasilopoulos A, Krska SW, Stahl SS. C(sp3)-H methylation enabled by peroxide photosensitization and Ni-mediated radical coupling. Science 2021;372:398-403. [PMID: 33888639 DOI: 10.1126/science.abh2623] [Cited by in Crossref: 13] [Cited by in F6Publishing: 4] [Article Influence: 13.0] [Reference Citation Analysis]
12 Gong PX, Xu F, Cheng L, Gong X, Zhang J, Gu WJ, Han W. Iron-catalyzed domino decarboxylation-oxidation of α,β-unsaturated carboxylic acids enabled aldehyde C-H methylation. Chem Commun (Camb) 2021;57:5905-8. [PMID: 34008616 DOI: 10.1039/d1cc01536b] [Reference Citation Analysis]
13 Rong X, Jin L, Gu Y, Liang G, Xia Q. Transition‐Metal‐Free Radical C−H Methylation of Quinoxalinones with TBHP. Asian J Org Chem 2020;9:185-8. [DOI: 10.1002/ajoc.201900758] [Cited by in Crossref: 9] [Cited by in F6Publishing: 3] [Article Influence: 4.5] [Reference Citation Analysis]
14 Lv W, Wen S, Liu J, Cheng G. Palladium-Catalyzed ortho -C–H Methylation of Benzoic Acids. J Org Chem 2019;84:9786-91. [DOI: 10.1021/acs.joc.9b01204] [Cited by in Crossref: 14] [Cited by in F6Publishing: 11] [Article Influence: 4.7] [Reference Citation Analysis]
15 Feng B, Yang Y, You J. A methylation platform of unconventional inert aryl electrophiles: trimethylboroxine as a universal methylating reagent. Chem Sci 2020;11:6031-5. [PMID: 34094095 DOI: 10.1039/d0sc01641a] [Cited by in Crossref: 10] [Article Influence: 5.0] [Reference Citation Analysis]
16 Sarki N, Goyal V, Natte K, Jagadeesh RV. Base Metal‐Catalyzed C‐Methylation Reactions Using Methanol. Adv Synth Catal 2021;363:5028-46. [DOI: 10.1002/adsc.202100762] [Cited by in Crossref: 1] [Article Influence: 1.0] [Reference Citation Analysis]
17 Steverlynck J, Sitdikov R, Rueping M. The Deuterated "Magic Methyl" Group: A Guide to Site-Selective Trideuteromethyl Incorporation and Labeling by Using CD3 Reagents. Chemistry 2021;27:11751-72. [PMID: 34076925 DOI: 10.1002/chem.202101179] [Cited by in Crossref: 1] [Cited by in F6Publishing: 1] [Article Influence: 1.0] [Reference Citation Analysis]
18 Koutoulogenis GS, Kokotou MG, Hayashi D, Mouchlis VD, Dennis EA, Kokotos G. 2-Oxoester Phospholipase A2 Inhibitors with Enhanced Metabolic Stability. Biomolecules 2020;10:E491. [PMID: 32213911 DOI: 10.3390/biom10030491] [Cited by in Crossref: 3] [Cited by in F6Publishing: 3] [Article Influence: 1.5] [Reference Citation Analysis]
19 Pan C, Yuan C, Yu JT. Peroxide-mediated synthesis of benzimidazo[2,1-a]isoquinoline-6(5H)-ones via cascade methylation/ethylation and intramolecular cyclization. Org Biomol Chem 2021;19:619-26. [PMID: 33367428 DOI: 10.1039/d0ob02383c] [Cited by in Crossref: 8] [Cited by in F6Publishing: 2] [Article Influence: 8.0] [Reference Citation Analysis]
20 Yang QL, Liu Y, Liang L, Li ZH, Qu GR, Guo HM. Facilitating Rh-Catalyzed C-H Alkylation of (Hetero)arenes and 6-Arylpurine Nucleosides (Nucleotides) with Electrochemistry. J Org Chem 2022. [PMID: 35438486 DOI: 10.1021/acs.joc.2c00391] [Reference Citation Analysis]
21 Lv W, Chen Y, Wen S, Ba D, Cheng G. Modular and Stereoselective Synthesis of C-Aryl Glycosides via Catellani Reaction. J Am Chem Soc 2020;142:14864-70. [PMID: 32808778 DOI: 10.1021/jacs.0c07634] [Cited by in Crossref: 17] [Cited by in F6Publishing: 6] [Article Influence: 8.5] [Reference Citation Analysis]
22 Kariofillis SK, Shields BJ, Tekle-Smith MA, Zacuto MJ, Doyle AG. Nickel/Photoredox-Catalyzed Methylation of (Hetero)aryl Chlorides Using Trimethyl Orthoformate as a Methyl Radical Source. J Am Chem Soc 2020;142:7683-9. [PMID: 32275411 DOI: 10.1021/jacs.0c02805] [Cited by in Crossref: 29] [Cited by in F6Publishing: 15] [Article Influence: 14.5] [Reference Citation Analysis]
23 Azeem Z, Mandal PK. Recent advances in palladium-catalyzed C(sp3)/C(sp2)-H bond functionalizations: access to C-branched glycosides. Org Biomol Chem 2022;20:264-81. [PMID: 34904995 DOI: 10.1039/d1ob02142g] [Reference Citation Analysis]
24 Jana R, Begam HM, Dinda E. The emergence of the C-H functionalization strategy in medicinal chemistry and drug discovery. Chem Commun (Camb) 2021;57:10842-66. [PMID: 34596175 DOI: 10.1039/d1cc04083a] [Reference Citation Analysis]
25 Ni S, Hribersek M, Baddigam SK, Ingner FJL, Orthaber A, Gates PJ, Pilarski LT. Mechanochemical Solvent‐Free Catalytic C−H Methylation. Angew Chem 2021;133:6734-40. [DOI: 10.1002/ange.202010202] [Cited by in Crossref: 8] [Cited by in F6Publishing: 5] [Article Influence: 4.0] [Reference Citation Analysis]
26 Ni S, Hribersek M, Baddigam SK, Ingner FJL, Orthaber A, Gates PJ, Pilarski LT. Mechanochemical Solvent-Free Catalytic C-H Methylation. Angew Chem Int Ed Engl 2021;60:6660-6. [PMID: 33031646 DOI: 10.1002/anie.202010202] [Cited by in Crossref: 15] [Cited by in F6Publishing: 8] [Article Influence: 7.5] [Reference Citation Analysis]
27 Shyni V, Leenaraj DR, Ittyachan R, Joseph L, Sajan D. Anticancer activity of indapamide adsorbed on gold nanoparticles: DFT, in-silico, and in-vitro analysis. J Mol Recognit 2021;34:e2920. [PMID: 34114274 DOI: 10.1002/jmr.2920] [Reference Citation Analysis]
28 Papeo G, Orsini P, Avanzi NR, Borghi D, Casale E, Ciomei M, Cirla A, Desperati V, Donati D, Felder ER, Galvani A, Guanci M, Isacchi A, Posteri H, Rainoldi S, Riccardi-Sirtori F, Scolaro A, Montagnoli A. Discovery of Stereospecific PARP-1 Inhibitor Isoindolinone NMS-P515. ACS Med Chem Lett 2019;10:534-8. [PMID: 30996792 DOI: 10.1021/acsmedchemlett.8b00569] [Cited by in Crossref: 8] [Cited by in F6Publishing: 6] [Article Influence: 2.7] [Reference Citation Analysis]
29 Sun LQ, Mull E, D'Andrea S, Zheng B, Hiebert S, Gillis E, Bowsher M, Kandhasamy S, Baratam VR, Puttaswamy S, Pulicharla N, Vishwakrishnan S, Reddy S, Trivedi R, Sinha S, Sivaprasad S, Rao A, Desai S, Ghosh K, Anumula R, Kumar A, Rajamani R, Wang YK, Fang H, Mathur A, Rampulla R, Zvyaga TA, Mosure K, Jenkins S, Falk P, Tagore DM, Chen C, Rendunchintala K, Loy J, Meanwell NA, McPhee F, Scola PM. Discovery of BMS-986144, a Third-Generation, Pan-Genotype NS3/4A Protease Inhibitor for the Treatment of Hepatitis C Virus Infection. J Med Chem 2020;63:14740-60. [PMID: 33226226 DOI: 10.1021/acs.jmedchem.0c01296] [Cited by in Crossref: 3] [Cited by in F6Publishing: 3] [Article Influence: 1.5] [Reference Citation Analysis]
30 Mao N, Ye Y, Zhuo X, Ye X, Xie T. Recent advances of the site-specific direct methylation on aromatic rings. Tetrahedron 2021;96:132402. [DOI: 10.1016/j.tet.2021.132402] [Cited by in Crossref: 1] [Cited by in F6Publishing: 1] [Article Influence: 1.0] [Reference Citation Analysis]
31 Aynetdinova D, Callens MC, Hicks HB, Poh CYX, Shennan BDA, Boyd AM, Lim ZH, Leitch JA, Dixon DJ. Installing the “magic methyl” – C–H methylation in synthesis. Chem Soc Rev 2021;50:5517-63. [DOI: 10.1039/d0cs00973c] [Cited by in Crossref: 17] [Cited by in F6Publishing: 2] [Article Influence: 17.0] [Reference Citation Analysis]
32 Gao Q, Shang Y, Song F, Ye J, Liu ZS, Li L, Cheng HG, Zhou Q. Modular Dual-Tasked C-H Methylation via the Catellani Strategy. J Am Chem Soc 2019;141:15986-93. [PMID: 31512477 DOI: 10.1021/jacs.9b07857] [Cited by in Crossref: 39] [Cited by in F6Publishing: 21] [Article Influence: 13.0] [Reference Citation Analysis]
33 Feng B, Zhang G, Feng X, Chen Y. Palladium-catalyzed decarbonylative methylation of aryl carboxylic acids. Org Chem Front . [DOI: 10.1039/d1qo01756j] [Reference Citation Analysis]
34 Bercher OP, Plunkett S, Mortimer TE, Watson MP. Deaminative Reductive Methylation of Alkylpyridinium Salts. Org Lett 2021;23:7059-63. [PMID: 34464140 DOI: 10.1021/acs.orglett.1c02458] [Cited by in Crossref: 1] [Article Influence: 1.0] [Reference Citation Analysis]