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For: Flick AC, Ding HX, Leverett CA, Kyne RE, Liu KK, Fink SJ, O’donnell CJ. Synthetic approaches to the 2014 new drugs. Bioorganic & Medicinal Chemistry 2016;24:1937-80. [DOI: 10.1016/j.bmc.2016.03.004] [Cited by in Crossref: 44] [Cited by in F6Publishing: 32] [Article Influence: 7.3] [Reference Citation Analysis]
Number Citing Articles
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10 Prasad V, Mishra N, Agrahari AK, Singh SK, Mohapatra PP, Tiwari VK. Cycloelimination-assisted Combinatorial Synthesis of Diverse Heterocyclic Scaffolds of Chemotherapeutic Values. COC 2019;23:768-808. [DOI: 10.2174/1385272823666190405145805] [Cited by in Crossref: 2] [Article Influence: 0.7] [Reference Citation Analysis]
11 Rajamanickam S, Sah C, Mir BA, Ghosh S, Sethi G, Yadav V, Venkataramani S, Patel BK. Bu 4 NI-Catalyzed, Radical-Induced Regioselective N -Alkylations and Arylations of Tetrazoles Using Organic Peroxides/Peresters. J Org Chem 2020;85:2118-41. [DOI: 10.1021/acs.joc.9b02875] [Cited by in Crossref: 10] [Cited by in F6Publishing: 4] [Article Influence: 5.0] [Reference Citation Analysis]
12 Flick AC, Ding HX, Leverett CA, Kyne RE, Liu KK-, Fink SJ, O’donnell CJ. Synthetic Approaches to the New Drugs Approved During 2015. J Med Chem 2017;60:6480-515. [DOI: 10.1021/acs.jmedchem.7b00010] [Cited by in Crossref: 62] [Cited by in F6Publishing: 42] [Article Influence: 12.4] [Reference Citation Analysis]
13 Raymer B, Bhattacharya SK. Lead-like Drugs: A Perspective: Miniperspective. J Med Chem 2018;61:10375-84. [DOI: 10.1021/acs.jmedchem.8b00407] [Cited by in Crossref: 24] [Cited by in F6Publishing: 19] [Article Influence: 6.0] [Reference Citation Analysis]
14 Pathania S, Kashyap N, Singh V, Shankar R, Kumar K, Rawal RK. Development and Recent Advancement of SGLT2 Inhibitors for the Treatment Regime of T2DM. J Biomed 2016;1. [DOI: 10.5812/jmb.10052] [Cited by in Crossref: 2] [Cited by in F6Publishing: 1] [Article Influence: 0.3] [Reference Citation Analysis]
15 Ayala-Aguilera CC, Valero T, Lorente-Macías Á, Baillache DJ, Croke S, Unciti-Broceta A. Small Molecule Kinase Inhibitor Drugs (1995-2021): Medical Indication, Pharmacology, and Synthesis. J Med Chem 2021. [PMID: 34624192 DOI: 10.1021/acs.jmedchem.1c00963] [Reference Citation Analysis]
16 Wang X, Sun H, Liu J, Zhong W, Zhang M, Zhou H, Dai D, Lu X. Palladium-Promoted DNA-Compatible Heck Reaction. Org Lett 2019;21:719-23. [DOI: 10.1021/acs.orglett.8b03926] [Cited by in Crossref: 32] [Cited by in F6Publishing: 28] [Article Influence: 10.7] [Reference Citation Analysis]
17 Flick AC, Leverett CA, Ding HX, Mcinturff E, Fink SJ, Helal CJ, O’donnell CJ. Synthetic Approaches to the New Drugs Approved During 2017. J Med Chem 2019;62:7340-82. [DOI: 10.1021/acs.jmedchem.9b00196] [Cited by in Crossref: 23] [Cited by in F6Publishing: 16] [Article Influence: 7.7] [Reference Citation Analysis]
18 Reig M, Bosque R, Font-bardía M, Calvis C, Messeguer R, Baldomà L, Badía J, Velasco D, López C. A study of the properties, reactivity and anticancer activity of novel N-methylated-3-thiazolyl or 3-thienyl carbazoles and their Pd(II) and Pt(II) complexes. Journal of Inorganic Biochemistry 2018;184:134-45. [DOI: 10.1016/j.jinorgbio.2018.03.008] [Cited by in Crossref: 3] [Cited by in F6Publishing: 2] [Article Influence: 0.8] [Reference Citation Analysis]
19 Pretelín-Castillo G, Silva Miranda M, Espitia C, Chávez-Santos RM, Suárez-Castro A, Chacón-García L, Aguayo-Ortiz R, Martinez R. (2Z)-3-Hydroxy-3-(4-R-Phenyl)-Prop-2-Enedithioic Acids as New Antituberculosis Compounds. Infect Drug Resist 2021;14:4323-32. [PMID: 34707377 DOI: 10.2147/IDR.S328132] [Reference Citation Analysis]
20 D'errico S, Borbone N, Piccialli V, Di Gennaro E, Zotti A, Budillon A, Vitagliano C, Piccialli I, Oliviero G. Synthesis and Evaluation of the Antitumor Properties of a Small Collection of Pt II Complexes with 7-Deazaadenosine as Scaffold: Synthesis and Evaluation of the Antitumor Properties of a Small Collection of Pt II Complexes with 7-Deazaadenosine as Scaffold. Eur J Org Chem 2017;2017:4935-47. [DOI: 10.1002/ejoc.201700730] [Cited by in Crossref: 6] [Cited by in F6Publishing: 3] [Article Influence: 1.2] [Reference Citation Analysis]
21 Zuo R, Zhang Y, Jiang C, Hackett JC, Loria R, Bruner SD, Ding Y. Engineered P450 biocatalysts show improved activity and regio-promiscuity in aromatic nitration. Sci Rep 2017;7:842. [PMID: 28405004 DOI: 10.1038/s41598-017-00897-z] [Cited by in Crossref: 18] [Cited by in F6Publishing: 18] [Article Influence: 3.6] [Reference Citation Analysis]
22 Xu F, Kim J, Waldman J, Wang T, Devine P. Synthesis of Grazoprevir, a Potent NS3/4a Protease Inhibitor for the Treatment of Hepatitis C Virus. Org Lett 2018;20:7261-5. [DOI: 10.1021/acs.orglett.8b03173] [Cited by in Crossref: 6] [Cited by in F6Publishing: 1] [Article Influence: 1.5] [Reference Citation Analysis]
23 Yu M, Lou S, Gonzalez-bobes F. Ring-Closing Metathesis in Pharmaceutical Development: Fundamentals, Applications, and Future Directions. Org Process Res Dev 2018;22:918-46. [DOI: 10.1021/acs.oprd.8b00093] [Cited by in Crossref: 43] [Cited by in F6Publishing: 11] [Article Influence: 10.8] [Reference Citation Analysis]
24 Zou L, Bennett R, Haidar Ahmad IA, Jocher BM, Zhang L, Bu X, Mangion I, Regalado EL. Generic Ion Chromatography–Conductivity Detection Method for Analysis of Palladium Scavengers in New Drug Substances. Org Process Res Dev 2019;23:1060-8. [DOI: 10.1021/acs.oprd.9b00101] [Cited by in Crossref: 8] [Cited by in F6Publishing: 7] [Article Influence: 2.7] [Reference Citation Analysis]
25 Wang S, Yuan XH, Wang SQ, Zhao W, Chen XB, Yu B. FDA-approved pyrimidine-fused bicyclic heterocycles for cancer therapy: Synthesis and clinical application. Eur J Med Chem 2021;214:113218. [PMID: 33540357 DOI: 10.1016/j.ejmech.2021.113218] [Cited by in Crossref: 3] [Cited by in F6Publishing: 2] [Article Influence: 3.0] [Reference Citation Analysis]
26 Liu J, Xu Y, Groszewicz PB, Brodrecht M, Fasel C, Hofmann K, Tan X, Gutmann T, Buntkowsky G. Novel dirhodium coordination polymers: the impact of side chains on cyclopropanation. Catal Sci Technol 2018;8:5190-200. [DOI: 10.1039/c8cy01493k] [Cited by in Crossref: 10] [Article Influence: 2.5] [Reference Citation Analysis]
27 Showalter HD. Recent Progress in the Discovery and Development of 2-Nitroimidazooxazines and 6-Nitroimidazooxazoles to Treat Tuberculosis and Neglected Tropical Diseases. Molecules 2020;25:E4137. [PMID: 32927749 DOI: 10.3390/molecules25184137] [Cited by in Crossref: 2] [Article Influence: 1.0] [Reference Citation Analysis]
28 Liu J, Sun B, Zhao X, Xing J, Gao Y, Chang W, Ji J, Zheng H, Cui C, Ji A, Lou H. Discovery of Potent Orally Active Protease-Activated Receptor 1 (PAR1) Antagonists Based on Andrographolide. J Med Chem 2017;60:7166-85. [DOI: 10.1021/acs.jmedchem.7b00951] [Cited by in Crossref: 11] [Cited by in F6Publishing: 7] [Article Influence: 2.2] [Reference Citation Analysis]
29 Khan S, Wang Y, Zhang M, Perveen S, Zhang J, Khan A. Regio- and enantioselective formation of tetrazole-bearing quaternary stereocenters via palladium-catalyzed allylic amination. Org Chem Front 2022;9:456-61. [DOI: 10.1039/d1qo01648b] [Cited by in Crossref: 1] [Cited by in F6Publishing: 1] [Article Influence: 1.0] [Reference Citation Analysis]
30 Flick AC, Leverett CA, Ding HX, McInturff E, Fink SJ, Mahapatra S, Carney DW, Lindsey EA, DeForest JC, France SP, Berritt S, Bigi-Botterill SV, Gibson TS, Liu Y, O'Donnell CJ. Synthetic Approaches to the New Drugs Approved during 2019. J Med Chem 2021;64:3604-57. [PMID: 33783211 DOI: 10.1021/acs.jmedchem.1c00208] [Cited by in Crossref: 2] [Cited by in F6Publishing: 1] [Article Influence: 2.0] [Reference Citation Analysis]
31 Phakhodee W, Duangkamol C, Wiriya N, Pattarawarapan M. Ultrasound-assisted synthesis of substituted 2-aminobenzimidazoles, 2-aminobenzoxazoles, and related heterocycles. Tetrahedron Letters 2016;57:5290-3. [DOI: 10.1016/j.tetlet.2016.10.060] [Cited by in Crossref: 15] [Cited by in F6Publishing: 7] [Article Influence: 2.5] [Reference Citation Analysis]
32 Ning XQ, Lou SJ, Mao YJ, Xu ZY, Xu DQ. Nitrate-promoted Selective C-H Fluorination of Benzamides and Benzeneacetamides. Org Lett 2018;20:2445-8. [PMID: 29634276 DOI: 10.1021/acs.orglett.8b00793] [Cited by in Crossref: 24] [Cited by in F6Publishing: 21] [Article Influence: 6.0] [Reference Citation Analysis]
33 Liu P, Zhang Z, Wang J, Zhang X, Yu X, Li Y. Empagliflozin protects diabetic pancreatic tissue from damage by inhibiting the activation of the NLRP3/caspase-1/GSDMD pathway in pancreatic β cells: in vitro and in vivo studies. Bioengineered 2021;12:9356-66. [PMID: 34823419 DOI: 10.1080/21655979.2021.2001240] [Reference Citation Analysis]
34 Hommelsheim R, Hock KJ, Schumacher C, Hussein MA, Nguyen TV, Koenigs RM. Cyanomethyl anion transfer reagents for diastereoselective Corey-Chaykovsky cyclopropanation reactions. Chem Commun (Camb) 2018;54:11439-42. [PMID: 30250960 DOI: 10.1039/c8cc05602a] [Cited by in Crossref: 7] [Cited by in F6Publishing: 1] [Article Influence: 1.8] [Reference Citation Analysis]
35 Martínez R, Espitia-Pinzón CI, Silva Miranda M, Chávez-Santos RM, Pretelin-Castillo G, Ramos-Orea A, Hernández-Báez ÁM, Cotlame-Pérez S, Pedraza-Rodríguez R. Synthesis and antituberculosis activity of new acylthiosemicarbazides designed by structural modification. Drug Dev Res 2020;81:350-5. [PMID: 31777976 DOI: 10.1002/ddr.21626] [Reference Citation Analysis]
36 Murata Y, Matsumoto N, Miyata M, Kitamura Y, Kakusawa N, Matsumura M, Yasuike S. One-pot reaction for the synthesis of N -substituted 2-aminobenzoxazoles using triphenylbismuth dichloride as cyclodesulfurization reagent. Journal of Organometallic Chemistry 2018;859:18-23. [DOI: 10.1016/j.jorganchem.2018.01.041] [Cited by in Crossref: 13] [Cited by in F6Publishing: 4] [Article Influence: 3.3] [Reference Citation Analysis]
37 Hock KJ, Spitzner R, Koenigs RM. Towards nitrile-substituted cyclopropanes – a slow-release protocol for safe and scalable applications of diazo acetonitrile. Green Chem 2017;19:2118-22. [DOI: 10.1039/c7gc00602k] [Cited by in Crossref: 35] [Article Influence: 7.0] [Reference Citation Analysis]
38 Hughes DL. Patent Review of Manufacturing Routes to Recently Approved PARP Inhibitors: Olaparib, Rucaparib, and Niraparib. Org Process Res Dev 2017;21:1227-44. [DOI: 10.1021/acs.oprd.7b00235] [Cited by in Crossref: 17] [Cited by in F6Publishing: 9] [Article Influence: 3.4] [Reference Citation Analysis]
39 Reilly SW, Mach RH. Pd-Catalyzed Synthesis of Piperazine Scaffolds Under Aerobic and Solvent-Free Conditions. Org Lett 2016;18:5272-5. [PMID: 27736075 DOI: 10.1021/acs.orglett.6b02591] [Cited by in Crossref: 27] [Cited by in F6Publishing: 16] [Article Influence: 4.5] [Reference Citation Analysis]
40 Gonçalves HA, Pereira BA, Teixeira WK, Moura S, Flores DC, Flores AF. Synthesis of 2,2,2-trifluoroethyl 1H-pyrazole carboxylates: Insight into the mechanism of trichloromethyl group hydrolysis. Journal of Fluorine Chemistry 2016;187:40-5. [DOI: 10.1016/j.jfluchem.2016.05.009] [Cited by in Crossref: 5] [Cited by in F6Publishing: 2] [Article Influence: 0.8] [Reference Citation Analysis]
41 Dhameliya TM, Donga HA, Vaghela PV, Panchal BG, Sureja DK, Bodiwala KB, Chhabria MT. A decennary update on applications of metal nanoparticles (MNPs) in the synthesis of nitrogen- and oxygen-containing heterocyclic scaffolds. RSC Adv 2020;10:32740-820. [DOI: 10.1039/d0ra02272a] [Cited by in Crossref: 6] [Article Influence: 3.0] [Reference Citation Analysis]
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