Review
Copyright ©The Author(s) 2015.
World J Virology. May 12, 2015; 4(2): 56-77
Published online May 12, 2015. doi: 10.5501/wjv.v4.i2.56
Table 1 Antiretroviral drugs class
Antiretroviral classGeneric name drugTrade name/manufacturer/approval (yr)
Nucleos(t)ide reverse transcriptase inhibitorsAbacavir (ABC)Ziagen® ViiV Healthcare (1998)
Didanozine (ddl)Videx® Bristol-Myers Squibb Co. (1991)
Emtricitabine (FTC)Emtriva® Gilead Sci. (2003)
Lamivudine (3TC)Epivir® GlaxoSmithKline (1995)
Stavudine (d4T)Zerit® Bristol-Myers Squibb Co. (1994)
Tenofovir (TDF)Viread® Gilead Sci. (2001)
Zidovudine (AZT)Retrovir® ViiV Healthcare (1987)
Zalcitabine (ddC)Hivid® Roche (1992)
Non-nucleoside reverse transcriptase inhibitorsDelavirdine (DLV)Rescriptor® Pfizer (1997)
Efavirenz (EFV)Sustiva® Bristol-Myers Squibb Co. (1998)
Stocrin® Merck Sharp, Dohme (1998)
Nevirapine (NVP)Viramune® Boehringer Ingelheim (1996)
Etravirine (ETR)Intelence® Janssen-Cilag (2008)
Rilpivirine (RPV)Edurant® Janssen-Cilag (2011)
Protease inhibitorsAmprenavirAgenerase® GlaxoSmithKline (1999)
AtazanavirReyataz® Bristol-Myers Squibb Co. (2003)
DarunavirPrezista® Janssen-Cilag (2006)
FosamprenavirLexiva® ViiV Healthcare (2003)
IndinavirCrixivan® Merck and Co. (1996)
LopinavirKaletra® Abbott (2000)
NelfinavirViracept® ViiV Healthcare (1997)
RitonavirNorvir® AbbVie Inc. (1996)
SaquinavirInvirase® Roche (1995)
TipranavirAptivus® Boehringer Ingelheim (2005)
Fusion inhibitorsEnfuvirtide, T-20Fuzeon® Hoffmann La Roche (2003)
Integrase strand transfer inhibitorsDolutegravir (DTG)Tivicay® GlaxoSmithKline (2013)
Elvitegravir (EVG)Stribild® Gilead Sci. (2012)
Raltegravir (RAL)Isentress® Merck and Co. (2007)
Entry inhibitors (CC chemokine receptor 5 antagonists)SelzentryMaraviroc® Pfizer (2007)